SCHEMBL8782844

SCHEMBL8782844

COc1ccc(CN(C)CCO)cc1OCc1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.73
CYP1A2 P05177 1/20 0.73
CYP3A4 P08684 1/20 0.73
CYP2D6 P10635 1/20 0.73
CYP2C9 P11712 1/20 0.73
BLM P54132 1/20 0.73
KMT2A Q03164 4/20 0.71
MEN1 O00255 3/20 0.71
MAPK1 P28482 1/20 0.53
HSD17B10 Q99714 1/20 0.53
ALDH1A1 P00352 1/20 0.53
BCHE P06276 3/20 0.51
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.50
ACHE P22303 2/20 0.49
SMPD1 P17405 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
OPRK1 P41145 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9416643 0.87 KDM4E (0.81) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28312736 0.81 KDM4E (0.64) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL12296058 0.81 BCHE (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3239903 0.81 BCHE (0.60) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL31361425 0.81 BCHE (0.60) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8728729 0.79 KDM4E (0.72) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL514870 0.78 KMT2A (0.82) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2060386 0.78 MAPK1 (0.63) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8734889 0.77 KDM4E (0.70) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
Bromide SCHEMBL20482559 0.76 MAPK1 (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0595995-B1 ARYLAMIDOALKYL- AND ARYLAMINOALKYL-N-HYDROXYUREA COMPOUNDS AND -N-HYDROXYFORMAMIDE DERIVATIVES HAVING LIPOXYGENASE INHIBITORY ACTIVITY ABBOTT LAB (US) 1997-01-15 EP disclosed
US-5514702-A Arylamidoalkyl-N-hydroxyurea compounds having lipoxygenase inhibitory activity ABBOTT LABORATORIES (US) 1996-05-07 US disclosed
US-5214204-A Inhibitors of biosynthesis of leukotrienes ABBOTT LABORATORIES (US) 1993-05-25 US disclosed