SCHEMBL8785240

SCHEMBL8785240

O=C(O)c1cn(C2CC2)c2c(C(F)(F)F)c(F)ccc2c1=O

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 7/20 0.54
TOP2B Q02880 7/20 0.54
ALDH1A1 P00352 4/20 0.46
POLB P06746 2/20 0.46
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
KDM4E B2RXH2 4/20 0.45
LMNA P02545 2/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
KCNH2 Q12809 4/20 0.44
GSK3B P49841 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8785244 0.85 TOP2A (0.39) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL8084266 0.85 TOP2A (0.64) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL8061657 0.84 TOP2A (0.61) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL4248696 0.84 TOP2A (0.39) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL143295 0.84 TOP2A (0.60) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL8927420 0.83 ADRB2 (0.51) TOP2ATOP2BALDH1A1KDM4ELMNA
SCHEMBL4248698 0.82 TOP2A (0.38) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL2081014 0.82 TOP2A (0.56) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL4482132 0.82 ALDH1A1 (0.58) TOP2ATOP2BALDH1A1POLBCHRM2
SCHEMBL4996474 0.81 TOP2A (0.46) TOP2ATOP2BALDH1A1POLBCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1097423-A Quinolone-and naphthyridonecarboxylic acid derivatives BAYER AG (DE) 1995-01-18 CN claimed
EP-0607825-A1 6-H-4-OXO-3-quinoline-carboxylic acids and their analogues as antibacterial agents BAYER AG (DE) 1994-07-27 EP claimed
US-5648567-A INTERMEDIATES FOR BACTERICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-07-15 US disclosed
EP-0607826-B1 Fluoro-trifluoromethylbenzoic acid derivatives BAYER AG (DE) 1997-05-07 EP disclosed
US-5493048-A REACTING METALLIZED FLUORO-TRIFLUOROMETHYLBENZENE DERIVATIVE WITH CARBON DIOXIDE AND PRODUCT IS THEN HYDROLYSED WITH AN ACID TO FORM ACID, SIMILARLY HALOGENATION GIVE ACID HALIDE AND WITH ALCOHOL GIVES ESTER BAYER AKTIENGESELLSCHAFT (DE) 1996-02-20 US disclosed
US-5457104-A Antibacterials BAYER AKTIENGESELLSCHAFT (DE) 1995-10-10 US disclosed
CN-1097423-A Quinolone-and naphthyridonecarboxylic acid derivatives BAYER AG (DE) 1995-01-18 CN disclosed
EP-0607826-A1 Fluoro-Trifluoromethylbenzoic acid derivatives BAYER AG (DE) 1994-07-27 EP disclosed
EP-0607825-A1 6-H-4-OXO-3-quinoline-carboxylic acids and their analogues as antibacterial agents BAYER AG (DE) 1994-07-27 EP disclosed