SCHEMBL8787553

SCHEMBL8787553

OCCCCN1CCC(c2onc3cc(F)ccc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.47
DRD2 P14416 4/20 0.47
SLC6A4 P31645 1/20 0.47
HTR2A P28223 4/20 0.46
KCNH2 Q12809 2/20 0.46
HTR7 P34969 1/20 0.46
HTR1A P08908 2/20 0.44
ADRA2A P08913 1/20 0.44
ADRA1D P25100 1/20 0.44
HTR2C P28335 1/20 0.44
ADRA1A P35348 1/20 0.44
HRH1 P35367 1/20 0.44
ADRA1B P35368 1/20 0.44
HTR6 P50406 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8787796 0.97 ACHE (0.48) ACHEDRD2SLC6A4HTR2AKCNH2
SCHEMBL8786866 0.92 ACHE (0.50) ACHEDRD2SLC6A4HTR2AKCNH2
SCHEMBL8788176 0.89 ACHE (0.47) ACHEDRD2SLC6A4HTR2AKCNH2
Hydrochloric Acid SCHEMBL8786999 0.88 ACHE (0.47) ACHEDRD2SLC6A4HTR2AKCNH2
SCHEMBL8787897 0.87 ACHE (0.48) ACHEDRD2SLC6A4HTR2AKCNH2
Hydrochloric Acid SCHEMBL8788247 0.86 ACHE (0.47) ACHEDRD2SLC6A4HTR2AKCNH2
SCHEMBL8506902 0.85 ACHE (0.50) ACHEDRD2SLC6A4HTR2AKCNH2
SCHEMBL8789014 0.84 HTR2A (0.53) DRD2HTR2AKCNH2HTR1AADRA2A
SCHEMBL8789335 0.83 ACHE (0.47) ACHEDRD2SLC6A4HTR2AKCNH2
SCHEMBL8871920 0.83 DRD2 (0.48) ACHEDRD2SLC6A4HTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP disclosed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP disclosed