Ilonidap

Ilonidap

SCHEMBL8788134

NC(=O)N1C(=O)C(=C(O)c2cccs2)c2cc(F)c(Cl)cc21.[Na]

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
KMT2A Q03164 3/20 0.34
RXFP1 Q9HBX9 3/20 0.34
KDM4E B2RXH2 2/20 0.34
POLB P06746 2/20 0.34
MAPT P10636 4/20 0.34
TDP1 Q9NUW8 3/20 0.33
MEN1 O00255 2/20 0.33
MAPK1 P28482 2/20 0.33
NOS1 P29475 1/20 0.33
PAX8 Q06710 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
HTT P42858 1/20 0.33
EGFR P00533 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ilonidap SCHEMBL8587853 0.99 ALDH1A1 (0.35) ALDH1A1KMT2ARXFP1KDM4EPOLB
Ilonidap SCHEMBL42518 0.99 ALDH1A1 (0.35) ALDH1A1KMT2ARXFP1KDM4EPOLB
Ilonidap SCHEMBL8587849 0.99 ALDH1A1 (0.35) ALDH1A1KMT2ARXFP1KDM4EPOLB
Ilonidap SCHEMBL8788348 0.98 ALDH1A1 (0.34) ALDH1A1KMT2ARXFP1KDM4EPOLB
Ilonidap SCHEMBL9284472 0.98 ALDH1A1 (0.34) ALDH1A1KMT2ARXFP1KDM4EPOLB
Ilonidap SCHEMBL8788132 0.98 ALDH1A1 (0.34) ALDH1A1KMT2ARXFP1KDM4EPOLB
SCHEMBL8788043 0.85 KMT2A (0.34) ALDH1A1KMT2ARXFP1KDM4EPOLB
SCHEMBL8788038 0.85 KMT2A (0.34) ALDH1A1KMT2ARXFP1KDM4EPOLB
SCHEMBL8787717 0.84 KMT2A (0.36) ALDH1A1KMT2ARXFP1KDM4EPOLB
SCHEMBL9449352 0.83 KDR (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0681580-B1 PRODRUGS OF ANTIINFLAMMATORY 3-ACYL-2-OXINDOLE-1-CARBOXAMIDES PFIZER (US) 1997-07-09 EP disclosed
EP-0681580-A1 PRODRUGS OF ANTIINFLAMMATORY 3-ACYL-2-OXINDOLE-1-CARBOXAMIDES. PFIZER HOSPITAL PROD (US) 1995-11-15 EP disclosed
WO-1994017061-A1 PRODRUGS OF ANTIINFLAMMATORY 3-ACYL-2-OXINDOLE-1-CARBOXAMIDES PFIZER INC. (US) 1994-08-04 WO disclosed
US-5270331-A Prodrugs of antiinflammatory 3-acyl-2-oxindole-1-carboxamides PFIZER, INC. (US) 1993-12-14 US disclosed