SCHEMBL8788424

SCHEMBL8788424

CCCNCCNc1ccc(NCCNCCC)c2c1C(=O)c1ccncc1C2=O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.63
MUS81 Q96NY9 1/20 0.63
TOP2B Q02880 1/20 0.51
BLM P54132 6/20 0.42
TP53 P04637 5/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
CYP3A4 P08684 4/20 0.42
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
MAPK1 P28482 3/20 0.42
USP2 O75604 2/20 0.42
LMNA P02545 2/20 0.42
RECQL P46063 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
NSD2 O96028 2/20 0.42
NPC1 O15118 2/20 0.42
MTOR P42345 2/20 0.42
RAB9A P51151 2/20 0.42
KDM6B O15054 2/20 0.42
KDM4C Q9H3R0 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8789454 0.90 ECE1 (0.58) ECE1MUS81TOP2BBLMTP53
SCHEMBL8788385 0.86 TOP2B (0.70) ECE1MUS81TOP2BBLMTP53
SCHEMBL8791572 0.86 ECE1 (0.51) ECE1MUS81TOP2BBLMTP53
SCHEMBL13035005 0.85 ECE1 (0.83) ECE1MUS81TOP2BBLMTP53
SCHEMBL8788938 0.85 ECE1 (0.57) ECE1MUS81TOP2BBLMTP53
Hydrochloric Acid SCHEMBL8788992 0.83 ECE1 (0.56) ECE1MUS81TOP2BBLMTP53
SCHEMBL8789103 0.82 ECE1 (0.55) ECE1MUS81TOP2BBLMTP53
SCHEMBL8791589 0.82 ECE1 (0.57) ECE1MUS81TOP2BBLMTP53
SCHEMBL8789428 0.81 ECE1 (0.62) ECE1MUS81TOP2BBLMTP53
SCHEMBL8788420 0.80 BLM (0.61) ECE1MUS81TOP2BBLMTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0503537-B1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones UNIV VERMONT (US) 1997-05-14 EP claimed
EP-0575526-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1993-12-29 EP claimed
WO-1992015300-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO[g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1992-09-17 WO claimed
EP-0503537-A1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones THE UNIVERSITY OF VERMONT (US) 1992-09-16 EP claimed
EP-0503537-B1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones UNIV VERMONT (US) 1997-05-14 EP disclosed
EP-0575526-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1993-12-29 EP disclosed
WO-1992015300-A1 6,9 BIS(SUBSTITUTED-AMINO)BENZO[g]ISOQUINOLINE-5,10-DIONES THE UNIVERSITY OF VERMONT (US) 1992-09-17 WO disclosed
EP-0503537-A1 6,9 Bis(substituted-amino)benzo-[g]isoquinoline-5,10-diones THE UNIVERSITY OF VERMONT (US) 1992-09-16 EP disclosed