SCHEMBL8788658

SCHEMBL8788658

COc1ccc(NC(C)=O)cc1OCCCN1CCC(c2onc3cc(F)ccc23)CC1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.60
HTR2A P28223 5/20 0.60
HTR1A P08908 4/20 0.60
ADRA2A P08913 3/20 0.60
HTR2C P28335 3/20 0.60
ADRA1A P35348 3/20 0.60
HRH1 P35367 3/20 0.60
HTR6 P50406 3/20 0.60
KCNH2 Q12809 3/20 0.60
ADRA1D P25100 2/20 0.60
ADRA1B P35368 2/20 0.60
ABCB11 O95342 1/20 0.56
CHRM2 P08172 1/20 0.56
CHRM1 P11229 1/20 0.56
ADRA2B P18089 1/20 0.56
ADRA2C P18825 1/20 0.56
DRD1 P21728 1/20 0.56
DRD4 P21917 1/20 0.56
ACHE P22303 1/20 0.56
SLC6A2 P23975 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8787873 0.87 DRD2 (0.63) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL458448 0.86 ABCB11 (0.74) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL8786884 0.86 DRD2 (0.58) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL1545101 0.86 HTR1A (0.78) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL8788442 0.85 DRD2 (0.58) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL8788937 0.85 HTR1A (0.53) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL8787916 0.84 HTR1A (0.51) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL5994919 0.84 HTR1A (0.69) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL8461799 0.84 HTR1A (0.52) DRD2HTR2AHTR1AADRA2AHTR2C
SCHEMBL8886291 0.84 ABCB11 (0.71) DRD2HTR2AHTR1AADRA2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663449-A FOR TREATING PSYCHOLOGICAL DISORDERS; ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1997-09-02 US disclosed
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP disclosed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP disclosed