SCHEMBL8790891

SCHEMBL8790891

COC(=O)CNC(=O)c1ccco1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.65
SMN1; SMN2 Q16637 3/20 0.65
TSHR P16473 2/20 0.62
KDM4E B2RXH2 2/20 0.59
PKM P14618 1/20 0.58
HSD17B10 Q99714 1/20 0.58
LMNA P02545 1/20 0.58
HPGD P15428 1/20 0.57
RAB9A P51151 3/20 0.55
NPC1 O15118 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
CYP1A2 P05177 1/20 0.54
CYP2C19 P33261 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12882119 0.86 ALDH1A1 (0.65) ALDH1A1SMN1; SMN2TSHRKDM4EPKM
SCHEMBL7926733 0.86 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2TSHRKDM4EPKM
SCHEMBL13074753 0.83 ALDH1A1 (0.64) ALDH1A1SMN1; SMN2KDM4EPKMHSD17B10
SCHEMBL13543194 0.82 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2TSHRKDM4EPKM
SCHEMBL237337 0.81 ALDH1A1 (0.66) ALDH1A1SMN1; SMN2TSHRPKMLMNA
SCHEMBL13545144 0.80 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2PKMHPGDRAB9A
SCHEMBL2969896 0.79 ALDH1A1 (0.64) ALDH1A1SMN1; SMN2PKMHPGDRAB9A
SCHEMBL4847926 0.79 ALDH1A1 (0.64) ALDH1A1SMN1; SMN2PKMHPGDRAB9A
SCHEMBL1232799 0.79 SMN1; SMN2 (0.75) ALDH1A1SMN1; SMN2PKMRAB9ANPC1
SCHEMBL11683297 0.79 ALDH1A1 (0.68) ALDH1A1SMN1; SMN2PKMHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4198029-A1 INHIBITORS OF PEPTIDYL ARGININE DEIMINASE (PAD) ENZYMES AND USES THEREOF University Health Network (CA) 2023-06-21 EP disclosed
WO-2017027967-A1 INHIBITORS OF PEPTIDYL ARGININE DEIMINASE (PAD) ENZYMES AND USES THEREOF UNIVERSITY HEALTH NETWORK (CA) 2017-02-23 WO disclosed
EP-0421365-B1 Tetrazoleacetic acid derivatives having aldose reductase inhibitory activity WAKAMOTO PHARMA CO LTD (JP) 1997-03-05 EP disclosed
US-RE35321-E ANTIDIABETIC AGENT WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1996-08-27 US disclosed
US-5068239-A Antidiabetic agent WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1991-11-26 US disclosed
EP-0421365-A2 Tetrazoleacetic acid derivatives having aldose reductase inhibitory activity Wakamoto Pharmaceutical Co., Ltd. (JP) 1991-04-10 EP disclosed