SCHEMBL8790959

SCHEMBL8790959

CC(=O)N1CCc2ccc(C(=O)CCCN3CCCCC3)cc2CC1

nearest known ligand 0.69

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 16/20 0.69
HRH3 Q9Y5N1 2/20 0.65
KDM4E B2RXH2 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8791256 0.84 ALDH1A1 (0.66) MCHR1HRH3KDM4E
SCHEMBL5432297 0.83 MCHR1 (0.62) MCHR1HRH3
SCHEMBL4850684 0.81 MCHR1 (0.61) MCHR1HRH3
SCHEMBL5423752 0.81 MCHR1 (1.00) MCHR1
SCHEMBL11679191 0.81 KDM4E (0.81) MCHR1HRH3KDM4EL3MBTL1
Hydrochloric Acid SCHEMBL11676911 0.80 KDM4E (0.79) MCHR1KDM4EL3MBTL1
Hydrochloric Acid SCHEMBL8790307 0.80 HTR1A (0.60) MCHR1KDM4EL3MBTL1
SCHEMBL11677718 0.79 KDM4E (0.79) MCHR1KDM4EL3MBTL1
SCHEMBL6071591 0.79 HRH3 (1.00) MCHR1HRH3
Trifluoroacetic Acid SCHEMBL6799476 0.78 MCHR1 (0.60) MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0560235-B1 Condensed heterocyclic ketone derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-06-04 EP disclosed
US-5462934-A Cholinesterase inhibitor; learning enhancement TAKEDA CHEMICAL INDUSTRIES (JP) 1995-10-31 US disclosed
EP-0560235-A1 Condensed heterocyclic ketone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-09-15 EP disclosed