SCHEMBL8790990

SCHEMBL8790990

CCOC(=O)CC(=O)c1ccc2c(c1)N(C(C)=O)CCCC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.52
ALDH1A1 P00352 6/20 0.48
LMNA P02545 2/20 0.48
HPGD P15428 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAPT P10636 3/20 0.47
HSD17B10 Q99714 1/20 0.47
OGG1 O15527 1/20 0.47
AVPR2 P30518 2/20 0.46
TSHR P16473 1/20 0.46
KDM4E B2RXH2 2/20 0.46
RECQL P46063 1/20 0.46
NOTUM Q6P988 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
OXTR P30559 1/20 0.41
AVPR1A P37288 1/20 0.41
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10856983 0.80 NOTUM (0.56) TP53ALDH1A1LMNAHPGDNPSR1
SCHEMBL8792645 0.79 NOTUM (0.56) TP53ALDH1A1LMNAHPGDAVPR2
SCHEMBL5418837 0.79 ALDH1A1 (0.49) TP53ALDH1A1LMNAHPGDMAPT
SCHEMBL5417050 0.77 ALDH1A1 (0.47) TP53ALDH1A1LMNAHPGDMAPT
SCHEMBL7487677 0.76 TP53 (0.52) TP53ALDH1A1LMNAHPGDNPSR1
SCHEMBL7488125 0.75 TP53 (0.44) TP53ALDH1A1LMNAHPGDNPSR1
SCHEMBL3082421 0.75 NOTUM (0.62) TP53ALDH1A1LMNAMAPTOGG1
SCHEMBL8791620 0.74 TP53 (0.43) TP53ALDH1A1LMNAHPGDNPSR1
SCHEMBL9206324 0.73 ACHE (0.58)
SCHEMBL15828391 0.72 ALDH1A1 (0.52) ALDH1A1LMNANPSR1MAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0560235-B1 Condensed heterocyclic ketone derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-06-04 EP disclosed
US-5462934-A Cholinesterase inhibitor; learning enhancement TAKEDA CHEMICAL INDUSTRIES (JP) 1995-10-31 US disclosed
EP-0560235-A1 Condensed heterocyclic ketone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-09-15 EP disclosed