SCHEMBL8793753

SCHEMBL8793753

CCOC(=O)c1[nH]c2c(C(F)(F)F)cccc2c1C(=O)OCC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
POLB P06746 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 2/20 0.44
HPGD P15428 2/20 0.44
ALOX5 P09917 4/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1252490 0.88 KDM4E (0.58) KDM4EPOLBALDH1A1GAAHPGD
SCHEMBL14829813 0.84 KDM4E (0.57) KDM4EPOLBCA12CA1CA2
SCHEMBL8795115 0.80 RXFP1 (0.62) CA12CA1CA2CA7CA9
SCHEMBL8794998 0.79 GAA (0.58) KDM4EPOLBCA12CA1CA2
SCHEMBL1998230 0.79 CA12 (0.59) KDM4EPOLBCA12CA1CA2
SCHEMBL31118679 0.78 KDM4E (0.64) KDM4EPOLBALDH1A1GAAHPGD
SCHEMBL10461607 0.76 KMT2A (0.51) KDM4EALDH1A1GAAHPGDALOX5
SCHEMBL22877825 0.76 KDM4E (0.58) KDM4EPOLBALOX5SMN1; SMN2PTGES
SCHEMBL10464236 0.74 ALOX15 (0.47) POLBCA12CA1CA2CA7
SCHEMBL13813425 0.74 SMN1; SMN2 (0.57) KDM4EPOLBALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0492485-B1 N-Acyl-2,3-benzodiazepine derivatives, pharmaceutical compositions containing them and process for preparing same GYOGYSZERKUTATO INTEZET (HU) 1997-11-19 EP claimed
US-5652239-A TREATMENT OF STROKES, ISCHEMIC ATTACK, ANTAGONISTS OF EXCITATORY AMINO ACIDS GLUTAMATE AND ASPARTATE IMPERIAL CHEMICAL COMPANY (GB) 1997-07-29 US disclosed
EP-0512817-B1 Pyridazinedione derivatives, their preparation and pharmaceutical applications ZENECA LTD (GB) 1997-02-19 EP disclosed
EP-0512817-A1 Pyridazinedione derivatives, their preparation and pharmaceutical applications ZENECA LIMITED (GB) 1992-11-11 EP disclosed