SCHEMBL8794022

SCHEMBL8794022

CC(C)N(C(=O)CN1C(=O)C(N)N=C(c2ccccc2)c2ccccc21)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.60
GABRP O00591 1/20 0.53
GABRD O14764 1/20 0.53
GABRA1 P14867 1/20 0.53
GABRB1 P18505 1/20 0.53
GABRG2 P18507 1/20 0.53
GABRB3 P28472 1/20 0.53
GABRA5 P31644 1/20 0.53
GABRA3 P34903 1/20 0.53
GABRA2 P47869 1/20 0.53
GABRB2 P47870 1/20 0.53
GABRA4 P48169 1/20 0.53
GABRE P78334 1/20 0.53
GABRA6 Q16445 1/20 0.53
GABRG1 Q8N1C3 1/20 0.53
GABRG3 Q99928 1/20 0.53
GABRQ Q9UN88 1/20 0.53
CCKAR P32238 8/20 0.51
CCKBR P32239 8/20 0.47
HDAC3 O15379 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8795033 0.99 ALDH1A1 (0.59) ALDH1A1GABRPGABRDGABRA1GABRB1
Bromide SCHEMBL8795037 0.99 ALDH1A1 (0.59) ALDH1A1GABRPGABRDGABRA1GABRB1
SCHEMBL8795883 0.88 ALDH1A1 (0.58) ALDH1A1CCKARCCKBRHDAC3HDAC1
SCHEMBL8796363 0.88 ALDH1A1 (0.62) ALDH1A1CCKARCCKBR
Bromide SCHEMBL8795194 0.87 ALDH1A1 (0.61) ALDH1A1CCKARCCKBR
SCHEMBL9573635 0.87 GABRP (0.56) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL9573630 0.85 GABRP (0.54) ALDH1A1GABRPGABRDGABRA1GABRB1
SCHEMBL9866449 0.83 CCKBR (0.61) ALDH1A1GABRPGABRDGABRA1GABRB1
SCHEMBL9867425 0.83 CCKBR (0.61) ALDH1A1GABRPGABRDGABRA1GABRB1
SCHEMBL9867431 0.83 CCKBR (0.61) ALDH1A1GABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755394-A1 A METHOD OF INDUCING CHOLECYSTOKININ AGONIST ACTIVITY USING 1,4-BENZODIAZEPINE COMPOUNDS GLAXO WELLCOME INC. (US) 1997-01-29 EP disclosed
WO-1995028399-A1 A METHOD OF INDUCING CHOLECYSTOKININ AGONIST ACTIVITY USING 1,4-BENZODIAZEPINE COMPOUNDS GLAXO WELLCOME INC. (US) 1995-10-26 WO disclosed