SCHEMBL8795162

SCHEMBL8795162

CCOC(=O)C1=CC(C)(C)Oc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
GSK3B P49841 1/20 0.45
CACNA1C Q13936 3/20 0.43
CACNA1F O60840 2/20 0.43
CACNA1D Q01668 2/20 0.43
CACNA1S Q13698 2/20 0.43
ADORA3 P0DMS8 2/20 0.43
MAPT P10636 4/20 0.42
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 3/20 0.41
PRKCZ Q05513 1/20 0.41
AR P10275 1/20 0.40
HIF1A Q16665 3/20 0.40
MEN1 O00255 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MAPK1 P28482 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6271007 0.86 SMN1; SMN2 (0.42) SMN1; SMN2GSK3BCACNA1CCACNA1FCACNA1D
Hydrochloric Acid SCHEMBL8796125 0.86 ALDH1A1 (0.37) SMN1; SMN2GSK3BCACNA1CCACNA1FCACNA1D
SCHEMBL8308734 0.82 AKR1B1 (0.43) MAPTALDH1A1KMT2AMEN1CYP3A4
SCHEMBL8794987 0.82 ALDH1A1 (0.36) SMN1; SMN2GSK3BCACNA1CCACNA1FCACNA1D
SCHEMBL8794980 0.82 ALDH1A1 (0.36) SMN1; SMN2GSK3BCACNA1CCACNA1FCACNA1D
SCHEMBL8794145 0.80 TP53 (0.38) MAPTALDH1A1KMT2AARCYP1A2
SCHEMBL8794716 0.79 MAPT (0.38) SMN1; SMN2MAPTALDH1A1KMT2AMEN1
SCHEMBL9566816 0.78 ALDH1A1 (0.41) MAPTALDH1A1KMT2AARHIF1A
SCHEMBL27328716 0.78 CA1 (0.38) MAPTALDH1A1KMT2AARMEN1
SCHEMBL27316930 0.78 PRSS1 (0.40) MAPTALDH1A1KMT2AARHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0541807-B1 NOVEL BENZOPYRAN DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 1997-12-17 EP disclosed
US-5412117-A Potassium channel activators, antiasmatics, antiepileptics CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 1995-05-02 US disclosed
EP-0541807-A1 NOVEL BENZOPYRAN DERIVATIVE Chugai Seiyaku Kabushiki Kaisha (JP) 1993-05-19 EP disclosed