SCHEMBL8795487

SCHEMBL8795487

CS(=O)(=O)O[C@H]1CC[C@H]([N+](=O)[O-])[C@@H](c2ccc(Cl)nc2)C1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 7/20 0.38
CHRNA4 P43681 7/20 0.38
CHRNA7 P36544 4/20 0.36
CHRNB4 P30926 3/20 0.36
CHRNA3 P32297 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
HPGD P15428 1/20 0.36
CHRND Q07001 1/20 0.36
CHRNA2 Q15822 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8977341 1.00 CHRNB2 (0.38) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL9235536 0.87 CHRNA7 (0.37) CHRNA7MEN1KMT2A
SCHEMBL9237968 0.86 MEN1 (0.35) MEN1KMT2A
SCHEMBL9240648 0.81 PTGS2 (0.34)
SCHEMBL8794532 0.81 KDM1A (0.42) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL8977318 0.81 KDM1A (0.42) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL8794944 0.79 CHRNB2 (0.45) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL8795614 0.79 CHRNB2 (0.45) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL6979465 0.78 CHRNB2 (0.39) CHRNB2CHRNA4CHRNA7CHRNB4CHRNA3
SCHEMBL9237183 0.75 DPP4 (0.36) ALDH1A1MEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657456-B1 Process for preparing epibatidine EGYT GYOGYSZERVEGYESZETI GYAR (HU) 1997-06-04 EP disclosed
EP-0657456-A1 Process for preparing epibatidine EGIS GYOGYSZERGYAR RT. (HU) 1995-06-14 EP disclosed
EP-0657455-A1 Epi-epibatidine derivatives, a process and intermediates for preparing them and epi-epibatidine and medicaments containing the epi-epibatidine derivatives and/or epi-epibatidine and the use of them EGIS GYOGYSZERGYAR (HU) 1995-06-14 EP disclosed