SCHEMBL8796103

SCHEMBL8796103

CCNc1cc2ncnc(NCc3cccc(OCCN4CCOCC4)c3)c2cc1[N+](=O)[O-]

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 6/20 0.56
RPS6KB1 P23443 6/20 0.56
ALDH1A1 P00352 2/20 0.44
USP2 O75604 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
PDGFRB P09619 1/20 0.44
EGFR P00533 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
PDPK1 O15530 1/20 0.43
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
HTT P42858 1/20 0.43
MAPT P10636 2/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8796911 0.96 AURKA (0.52) AURKARPS6KB1ALDH1A1USP2CYP1A2
SCHEMBL8796055 0.92 RPS6KB1 (0.47) AURKARPS6KB1ALDH1A1PDGFRBEGFR
SCHEMBL8796031 0.92 AURKA (0.48) AURKARPS6KB1ALDH1A1PDGFRBEGFR
SCHEMBL8795496 0.88 AURKA (0.49) AURKARPS6KB1ALDH1A1PDGFRBEGFR
SCHEMBL8796758 0.87 AURKA (0.44) AURKARPS6KB1ALDH1A1USP2CYP1A2
SCHEMBL8795542 0.87 AURKA (0.47) AURKARPS6KB1ALDH1A1PDGFRBEGFR
SCHEMBL8796285 0.85 SRC (0.47) USP2CYP1A2CYP3A4CYP2D6CLK4
SCHEMBL8795332 0.85 HTT (0.48) AURKARPS6KB1ALDH1A1USP2CYP1A2
SCHEMBL7525212 0.84 MAPT (0.52) AURKAALDH1A1PDGFRBEGFRSMN1; SMN2
SCHEMBL8796096 0.84 RPS6KB1 (0.46) AURKARPS6KB1ALDH1A1PDGFRBEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5698560-A TREATMENT OF CARDIOVASCULAR DISORDERS; ANTICOAGULANTS; CARDIOTONIC AGENTS; HYPOTENSIVE AGENTS; ARTERIOSCLEROSIS; CYCLIC GMP-SPECIFIC PHOSPHODIESTERASE INHIBITORS KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-12-16 US disclosed
EP-0758653-A1 IMIDAZOQUINAZOLINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-02-19 EP disclosed