SCHEMBL8796758

SCHEMBL8796758

CCNc1cc2ncnc(NCc3cccc(CN4CCOCC4)c3)c2cc1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.44
RPS6KB1 P23443 3/20 0.44
EGFR P00533 6/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
PDGFRB P09619 1/20 0.42
AURKB Q96GD4 1/20 0.41
KCNH2 Q12809 1/20 0.41
USP2 O75604 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
MET P08581 1/20 0.40
POLB P06746 1/20 0.40
MCL1 Q07820 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8796603 0.92 LMNA (0.44) EGFRMAPTALDH1A1L3MBTL1TDP1
SCHEMBL7525212 0.88 MAPT (0.52) AURKAEGFRMAPTALDH1A1L3MBTL1
SCHEMBL8796308 0.88 EGFR (0.47) EGFRMAPTALDH1A1L3MBTL1TDP1
SCHEMBL8796103 0.87 AURKA (0.56) AURKARPS6KB1EGFRMAPTALDH1A1
SCHEMBL8796911 0.87 AURKA (0.52) AURKARPS6KB1EGFRALDH1A1PDGFRB
SCHEMBL7523791 0.84 MAPT (0.53) EGFRMAPTALDH1A1L3MBTL1TDP1
SCHEMBL8796240 0.84 EGFR (0.45) EGFRMAPTALDH1A1PDGFRBCYP1A2
SCHEMBL8796234 0.84 PIK3CA (0.45) EGFRMAPTPDGFRBCYP1A2
SCHEMBL8795595 0.83 EGFR (0.49) EGFRPDGFRBCLK4
SCHEMBL8796541 0.83 EGFR (0.47) EGFRMAPTALDH1A1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5698560-A TREATMENT OF CARDIOVASCULAR DISORDERS; ANTICOAGULANTS; CARDIOTONIC AGENTS; HYPOTENSIVE AGENTS; ARTERIOSCLEROSIS; CYCLIC GMP-SPECIFIC PHOSPHODIESTERASE INHIBITORS KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-12-16 US disclosed
EP-0758653-A1 IMIDAZOQUINAZOLINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-02-19 EP disclosed