SCHEMBL8796181

SCHEMBL8796181

CC1(C)C=C(c2ccccn2)c2cc(OC(F)F)ccc2O1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.35
MAPT P10636 2/20 0.34
TSHR P16473 1/20 0.34
GAA P10253 1/20 0.34
CBFB Q13951 1/20 0.34
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP2E1 P05181 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C8 P10632 1/20 0.33
CYP2B6 P20813 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.32
BACE1 P56817 2/20 0.32
CTSD P07339 1/20 0.32
PTPN1 P18031 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8794576 0.86 CBFB (0.43) CBFB
SCHEMBL9524858 0.83 MAPT (0.37) MAPTTSHRGAACYP2C9CYP3A4
SCHEMBL8794694 0.80 RARA (0.38) CYP3A4BACE1CTSDKDM4ERECQL
SCHEMBL9527612 0.79 NPC1 (0.44) MAPTGAACBFBCYP1A2NPC1
SCHEMBL8795574 0.79 HSD17B10 (0.36) MAPTGAACYP1A2CYP2D6CYP2C9
SCHEMBL9524965 0.78 ADRA1A (0.39) MAPTCYP1A2NPC1RAB9ASMN1; SMN2
SCHEMBL9523928 0.78 CBFB (0.40) MAPTGAACBFBNPC1RAB9A
SCHEMBL9525700 0.77 KDM4E (0.39) MAPTGAACYP1A2CYP2D6CYP2C9
SCHEMBL9524854 0.77 RARA (0.48) KDM4ERARARARBRARG
SCHEMBL9525024 0.77 RARA (0.41) TSHRNPC1RAB9ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0586405-B1 NOVEL 2H-BENZO[b]PYRANE DERIVATIVES SUBSTITUTED IN THE 4 POSITION BY ARYL OR N-HETEROARYL, PROCESS FOR PRODUCING THEM AND PREPARATIONS CONTAINING THE COMPOUNDS BEIERSDORF LILLY GMBH (DE) 1997-09-10 EP disclosed
EP-0586405-A1 NOVEL 2H-BENZO b]PYRANE DERIVATIVES SUBSTITUTED IN THE 4 POSITION BY ARYL OR N-HETEROARYL, PROCESS FOR PRODUCING THEM AND PREPARATIONS CONTAINING THE COMPOUNDS. BEIERSDORF LILLY GMBH (DE) 1994-03-16 EP disclosed
WO-1992020671-A1 NOVEL 2H-BENZO[b]PYRANE DERIVATIVES SUBSTITUTED IN THE 4 POSITION BY ARYL OR N-HETEROARYL, PROCESS FOR PRODUCING THEM AND PREPARATIONS CONTAINING THE COMPOUNDS BEIERSDORF-LILLY GMBH (DE) 1992-11-26 WO disclosed