SCHEMBL8796643

SCHEMBL8796643

Cc1c[nH]c(-c2ccc(Br)c(C)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMP P19971 1/20 0.46
S1PR1 P21453 1/20 0.35
MAPT P10636 5/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HAO1 Q9UJM8 1/20 0.33
TSHR P16473 2/20 0.32
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP3A4 P08684 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
TDO2 P48775 1/20 0.31
CCNT1 O60563 1/20 0.31
PIM1 P11309 1/20 0.31
CDK9 P50750 1/20 0.31
HASPIN Q8TF76 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27985279 0.79 MAPK1 (0.40) TYMPMAPTALDH1A1NPC1PKM
SCHEMBL797826 0.78 TNKS (0.40) TYMPMAPTALDH1A1NPC1RAB9A
SCHEMBL12581386 0.76 ALDH1A1 (0.50) TYMPMAPTALDH1A1KDM4ENPC1
SCHEMBL29724664 0.74 CYP11B1 (0.45) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL535698 0.74 CYP11B1 (0.45) MAPTALDH1A1KDM4ENPC1RAB9A
SCHEMBL6647087 0.74 NISCH (0.48) TYMPMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL156929 0.72 TYMP (0.40) TYMPS1PR1MAPTALDH1A1KDM4E
SCHEMBL30949496 0.72 TDP2 (0.33)
SCHEMBL29522030 0.72 TYMP (0.40) TYMPS1PR1MAPTALDH1A1KDM4E
SCHEMBL7832944 0.72 NISCH (0.58) TYMPS1PR1ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799226-A1 TETRACYCLIC SPIRO COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THEIR USE AS 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-10-08 EP disclosed