SCHEMBL8796789

SCHEMBL8796789

O=C(CC(C(=O)O)c1nc(-c2ccc(-c3ccccc3)cc2)c[nH]1)OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.42
ROCK2 O75116 1/20 0.41
SLC15A1 P46059 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MAPK1 P28482 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PPARG P37231 6/20 0.37
PPARA Q07869 4/20 0.37
MCL1 Q07820 1/20 0.37
ROCK1 Q13464 1/20 0.36
MYLK4 Q86YV6 1/20 0.36
TSHR P16473 1/20 0.36
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797492 0.93 ENPP2 (0.42) ENPP2ROCK2SLC15A1SMN1; SMN2MAPK1
SCHEMBL8797073 0.91 ALDH1A1 (0.41) ENPP2ROCK2SLC15A1SMN1; SMN2MAPK1
SCHEMBL8798522 0.84 DHODH (0.45) SMN1; SMN2MAPK1L3MBTL1ALDH1A1PPARG
SCHEMBL14525072 0.84 SLC15A1 (0.44) ENPP2ROCK2SLC15A1SMN1; SMN2MAPK1
SCHEMBL14268347 0.84 SLC15A1 (0.44) ENPP2ROCK2SLC15A1SMN1; SMN2MAPK1
SCHEMBL14268348 0.84 SLC15A1 (0.44) ENPP2ROCK2SLC15A1SMN1; SMN2MAPK1
SCHEMBL394264 0.79 CPA1 (0.49) CYP1A2PPARGPPARA
SCHEMBL14268346 0.75 KLK7 (0.47) PPARGPPARAMEN1KMT2A
SCHEMBL14268345 0.75 KLK7 (0.47) PPARGPPARAMEN1KMT2A
SCHEMBL392816 0.74 TACR3 (0.47) ALDH1A1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0807114-A1 BRIDGED INDOLES AS MATRIX METALLOPROTEASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1997-11-19 EP disclosed