SCHEMBL8797161

SCHEMBL8797161

Cc1cc(C)nc(NCC(=O)NCC(N)=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.46
ALDH1A1 P00352 2/20 0.43
TP53 P04637 1/20 0.43
NOS3 P29474 1/20 0.42
NOS2 P35228 1/20 0.42
LCK P06239 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
SYK P43405 5/20 0.39
KCNH2 Q12809 4/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
GBA1 P04062 1/20 0.39
RAB9A P51151 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
SORT1 Q99523 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797859 0.99 MAPK1 (0.45) MAPK1ALDH1A1TP53NOS3NOS2
SCHEMBL8797444 0.89 NOS3 (0.48) MAPK1ALDH1A1TP53NOS3NOS2
SCHEMBL8797408 0.79 MAPK1 (0.46) MAPK1ALDH1A1TP53NOS3NOS2
SCHEMBL6508707 0.71 KMT2A (0.60) MAPK1ALDH1A1NOS3NOS2LCK
SCHEMBL8797441 0.70 MAPK1 (0.63) MAPK1ALDH1A1TP53NOS3NOS2
SCHEMBL8798095 0.70 MAPK1 (0.70) MAPK1ALDH1A1TP53NOS3NOS2
SCHEMBL8347190 0.69 KDM4E (0.63) MAPK1ALDH1A1TP53NOS3NOS2
SCHEMBL12182431 0.68 MAPK1 (0.65) MAPK1ALDH1A1TP53NOS3NOS2
SCHEMBL8345724 0.68 NOS3 (0.59) MAPK1ALDH1A1TP53NOS3NOS2
SCHEMBL7797450 0.67 NOS3 (0.53) MAPK1ALDH1A1TP53NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632026-B1 Alpha amino acid derivatives, a method for their preparation and pharmaceutical preparations containing them ADIR (FR) 1997-11-19 EP claimed
US-5470864-A Glycine amide derivatives containing pyridine or pyridine-N-oxide, anticholesterol, antiinflammatory ADIR ET COMPAGNIE (FR) 1995-11-28 US claimed
EP-0811001-A1 BENZOTHIAZINE DIOXIDES AS ENDOTHELIN ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1997-12-10 EP disclosed
EP-0632026-B1 Alpha amino acid derivatives, a method for their preparation and pharmaceutical preparations containing them ADIR (FR) 1997-11-19 EP disclosed
US-5585390-A ANTIINFLAMMATORY AGENTS; ANTILIPEMIC AGENTS ADIR ET COMPAGNIE (FR) 1996-12-17 US disclosed
US-5470864-A Glycine amide derivatives containing pyridine or pyridine-N-oxide, anticholesterol, antiinflammatory ADIR ET COMPAGNIE (FR) 1995-11-28 US disclosed
EP-0632026-A1 Alpha amino acid derivatives, a method for their preparation and pharmaceutical preparations containing them ADIR ET COMPAGNIE (FR) 1995-01-04 EP disclosed