SCHEMBL7797450

SCHEMBL7797450

Cc1cc(C)nc(NCCN)c1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.53
NOS2 P35228 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.51
TLR8 Q9NR97 1/20 0.45
NPY1R P25929 1/20 0.43
SYK P43405 1/20 0.43
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NOS1 P29475 1/20 0.42
KARS1 Q15046 1/20 0.41
MAPK1 P28482 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LCK P06239 1/20 0.39
IDH1 O75874 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12963699 0.82 NOS3 (0.55) NOS3NOS2SMN1; SMN2TLR8ALDH1A1
SCHEMBL15286809 0.81 SMN1; SMN2 (0.43) NOS3NOS2SMN1; SMN2TLR8NPY1R
SCHEMBL23482212 0.81 GAA (0.56) NOS3NOS2TLR8ALDH1A1MEN1
SCHEMBL9313985 0.79 TLR8 (0.65) NOS3NOS2SMN1; SMN2TLR8ALDH1A1
SCHEMBL15286764 0.79 SMN1; SMN2 (0.41) SMN1; SMN2TLR8NPY1RSYKKARS1
SCHEMBL15286470 0.79 SMN1; SMN2 (0.44) SMN1; SMN2TLR8SYKALDH1A1MEN1
SCHEMBL11187910 0.78 DNM2 (0.55) NOS3NOS2TLR8ALDH1A1NOS1
SCHEMBL24672584 0.78 TLR8 (0.58) NOS3NOS2SMN1; SMN2TLR8ALDH1A1
SCHEMBL9884955 0.78 SMN1; SMN2 (0.49) SMN1; SMN2TLR8NPY1RSYKALDH1A1
SCHEMBL8345724 0.78 NOS3 (0.59) NOS3NOS2SMN1; SMN2TLR8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0796847-B1 Pyridine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO CO LTD (JP) 2001-11-28 EP disclosed
US-6017937-A BACTERICIDE AGAINST HELICOBACTER PYROLI; INHIBITING ACID SECRETION IN STOMACH OF MAN OR MAMMALS, PREVENTING OR CURING ULCER SHISEIDO CO., LTD. (JP) 2000-01-25 US disclosed
US-5859032-A HAVING ANTIBACTERIAL ACTIVITY AGAINST HELICOBACTER PYLORI SHISEIDO CO., LTD. (JP) 1999-01-12 US disclosed
EP-0796847-A1 Pyridine derivative, anti-ulcer drug, and antibacterial drug SHISEIDO COMPANY LIMITED (JP) 1997-09-24 EP disclosed