SCHEMBL8797303

SCHEMBL8797303

COc1cccc2c1N(c1ccccc1)CN(CCOc1ccc(CC3NC(=O)SC3=O)cc1)C2=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.37
BCHE P06276 3/20 0.35
ACHE P22303 3/20 0.35
RAB9A P51151 2/20 0.34
UGCG Q16739 3/20 0.34
FFAR1 O14842 2/20 0.33
NPC1 O15118 1/20 0.33
ATM Q13315 1/20 0.33
MMP1 P03956 1/20 0.33
MMP3 P08254 1/20 0.33
MMP9 P14780 1/20 0.33
KCNH2 Q12809 1/20 0.33
TSHR P16473 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
OPRK1 P41145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8796692 0.96 HRH3 (0.40) HRH3BCHEACHEUGCGMMP1
SCHEMBL8803024 0.86 HRH3 (0.41) HRH3RAB9AFFAR1NPC1
SCHEMBL8797295 0.85 FFAR1 (0.49) HRH3FFAR1TSHRMEN1ALDH1A1
SCHEMBL8796714 0.82 ALDH1A1 (0.41) HRH3RAB9AFFAR1MEN1ALDH1A1
SCHEMBL8796685 0.81 HRH3 (0.49) HRH3FFAR1TSHRMEN1ALDH1A1
SCHEMBL8796706 0.81 HRH3 (0.38) HRH3BCHEACHEFFAR1ALDH1A1
SCHEMBL8796905 0.76 HRH3 (0.38) HRH3BCHEACHEKCNH2
SCHEMBL8799698 0.76 HRH3 (0.41) HRH3FFAR1
SCHEMBL8796863 0.76 HRH3 (0.35) HRH3BCHEACHEFFAR1KCNH2
SCHEMBL8797065 0.75 HRH3 (0.41) HRH3RAB9AFFAR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787727-A1 Benzoazine derivative or salt thereof and pharmaceutical composition comprising the same SS Pharmaceutical Co., Ltd. (JP) 1997-08-06 EP disclosed