SCHEMBL8797442

SCHEMBL8797442

c1ccc(-c2coc(-c3ccc[nH]3)c2-c2ccccc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.38
CSF1R P07333 2/20 0.36
MAPT P10636 1/20 0.32
ERCC5 P28715 2/20 0.31
FEN1 P39748 2/20 0.31
KDR P35968 2/20 0.31
AURKA O14965 1/20 0.31
PIN1 Q13526 1/20 0.30
IKBKB O14920 1/20 0.30
CHUK O15111 1/20 0.30
DAPK3 O43293 1/20 0.30
JAK2 O60674 1/20 0.30
PRKD3 O94806 1/20 0.30
MAP4K4 O95819 1/20 0.30
PAK4 O96013 1/20 0.30
RET P07949 1/20 0.30
IGF1R P08069 1/20 0.30
FGFR1 P11362 1/20 0.30
PRKACA P17612 1/20 0.30
FLT1 P17948 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797839 0.86 CSF1R (0.36) ADORA2ACSF1RMAPTKDRAURKA
SCHEMBL25706159 0.81 MAPT (0.39) MAPTPIN1ALDH1A1ALOX15HSD17B10
SCHEMBL24818258 0.79 ALDH1A1 (0.40) MAPTPIN1ALDH1A1ALOX15HSD17B10
SCHEMBL24817429 0.73 GPR84 (0.38) MAPTPIN1ALDH1A1ALOX15HSD17B10
SCHEMBL12469844 0.71 ADORA2A (0.44) ADORA2ACSF1RMAPTKDRAURKA
SCHEMBL80142 0.70 HDAC1 (0.48) ADORA2ACSF1RMAPTALDH1A1
SCHEMBL21806653 0.69 ADORA2A (0.43) ADORA2ACSF1RMAPTKDRAURKA
SCHEMBL28212557 0.68 HDAC1 (0.47) ADORA2ACSF1RMAPTKDRALDH1A1
SCHEMBL27515517 0.68 HDAC1 (0.47) ADORA2ACSF1RMAPTKDRALDH1A1
Fluoride SCHEMBL30394298 0.68 HDAC1 (0.47) ADORA2ACSF1RMAPTKDRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0597291-B1 2,3-diphenyl-5-pyrrolyl-furan derivatives, processes and intermediates for their preparation and their use as anti-inflammatory, and anti-allergic and platelet aggregation inhibiting agents NIHON IYAKUHIN KOGYO CO LTD (JP) 1997-06-11 EP claimed
US-5321041-A Antiallergens, antiinflammatory and anticaogulants NIHON IYAKUHIN KOGYO CO., LTD. (JP) 1994-06-14 US claimed
EP-0597291-A1 2,3-diphenyl-5-pyrrolyl-furan derivatives, processes and intermediates for their preparation and their use as anti-inflammatory, and anti-allergic and platelet aggregation inhibiting agents NIHON IYAKUHIN KOGYO CO., LTD. (JP) 1994-05-18 EP claimed
EP-0597291-B1 2,3-diphenyl-5-pyrrolyl-furan derivatives, processes and intermediates for their preparation and their use as anti-inflammatory, and anti-allergic and platelet aggregation inhibiting agents NIHON IYAKUHIN KOGYO CO LTD (JP) 1997-06-11 EP disclosed
US-5321041-A Antiallergens, antiinflammatory and anticaogulants NIHON IYAKUHIN KOGYO CO., LTD. (JP) 1994-06-14 US disclosed
US-5321041-A Antiallergens, antiinflammatory and anticaogulants NIHON IYAKUHIN KOGYO CO., LTD. (JP) 1994-06-14 US disclosed
EP-0597291-A1 2,3-diphenyl-5-pyrrolyl-furan derivatives, processes and intermediates for their preparation and their use as anti-inflammatory, and anti-allergic and platelet aggregation inhibiting agents NIHON IYAKUHIN KOGYO CO., LTD. (JP) 1994-05-18 EP disclosed
EP-0597291-A1 2,3-diphenyl-5-pyrrolyl-furan derivatives, processes and intermediates for their preparation and their use as anti-inflammatory, and anti-allergic and platelet aggregation inhibiting agents NIHON IYAKUHIN KOGYO CO., LTD. (JP) 1994-05-18 EP disclosed