SCHEMBL8798071

SCHEMBL8798071

COc1cc(Br)c(O)c(CBr)c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.47
PTGS2 P35354 1/20 0.47
ALOX15 P16050 1/20 0.41
ALOX12 P18054 1/20 0.41
CALM1 P0DP23 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ABL1 P00519 2/20 0.39
BCR P11274 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PTPN1 P18031 2/20 0.38
CYP1A2 P05177 1/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
RECQL P46063 1/20 0.37
RIN1 Q13671 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7642548 0.90 ALDH1A1 (0.43) CALM1CA1CA2ABL1BCR
SCHEMBL8797591 0.84 ALOX5 (0.47) ALOX5PTGS2ALOX15ALOX12CALM1
SCHEMBL30679916 0.84 ALOX5 (0.47) ALOX5PTGS2ALOX15ALOX12CALM1
SCHEMBL8797818 0.82 ALOX5 (0.46) ALOX5PTGS2ALOX15ALOX12CALM1
SCHEMBL28173580 0.81 CA1 (0.37) CALM1CA1CA2ABL1CYP3A4
SCHEMBL1119249 0.80 ALOX5 (0.54) ALOX5PTGS2ALOX15ALOX12CA1
SCHEMBL6827911 0.79 ALDH1A1 (0.46) CA2CYP3A4ALDH1A1CYP1A2
SCHEMBL6443831 0.78 ERN1 (0.42) ALOX5PTGS2ALOX15ALOX12CALM1
SCHEMBL31488167 0.78 CA2 (0.67) PTGS2ALOX15CA1CA2CYP3A4
SCHEMBL957652 0.78 CYP3A4 (0.40) CYP3A4ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0542671-B1 Substituted hydroquinone derivatives as intermediates of benzofuran derivatives CIBA GEIGY AG (CH) 1997-01-02 EP claimed
EP-0542671-A1 Substituted hydroquinone derivatives as intermediates of benzofuran derivatives CIBA-GEIGY AG (CH) 1993-05-19 EP claimed
US-5693807-A Substituted hydroquinone derivatives CIBA-GEIGY CORPORATION (US) 1997-12-02 US disclosed
EP-0542671-B1 Substituted hydroquinone derivatives as intermediates of benzofuran derivatives CIBA GEIGY AG (CH) 1997-01-02 EP disclosed
US-5290939-A Process for the manufacture of brofaromine and analogs thereof CIBA-GEIGY CORPORATION (US) 1994-03-01 US disclosed
EP-0542671-A1 Substituted hydroquinone derivatives as intermediates of benzofuran derivatives CIBA-GEIGY AG (CH) 1993-05-19 EP disclosed