SCHEMBL8798290

SCHEMBL8798290

c1ccc(Nc2cc(N3CCCC3)ncn2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.59
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
TSHR P16473 1/20 0.55
RECQL P46063 1/20 0.55
CD274 Q9NZQ7 1/20 0.54
HRH4 Q9H3N8 2/20 0.52
PIK3CB P42338 1/20 0.52
ABL1 P00519 1/20 0.50
BCR P11274 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
SCN9A Q15858 1/20 0.47
POLB P06746 1/20 0.47
ALDH1A1 P00352 2/20 0.47
ATM Q13315 1/20 0.47
LMNA P02545 2/20 0.46
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
MAPK10 P53779 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31660945 0.98 SMN1; SMN2 (0.61) SMN1; SMN2NPC1RAB9ATSHRRECQL
SCHEMBL31660951 0.88 CD274 (0.51) SMN1; SMN2NPC1RAB9ATSHRCD274
SCHEMBL27330852 0.87 ABL1 (0.66) NPC1RAB9ARECQLPIK3CBABL1
SCHEMBL14421264 0.85 CD274 (0.55) SMN1; SMN2NPC1RAB9ATSHRRECQL
SCHEMBL27741343 0.85 CD274 (0.55) SMN1; SMN2NPC1RAB9ATSHRRECQL
SCHEMBL27332171 0.84 ADORA3 (0.53) SMN1; SMN2RAB9ACD274SCN9AALDH1A1
SCHEMBL27334586 0.84 SMN1; SMN2 (0.62) SMN1; SMN2NPC1RAB9ACD274ABL1
SCHEMBL14421382 0.82 CCNE1 (0.56) SMN1; SMN2NPC1RAB9ATSHRRECQL
SCHEMBL27318007 0.81 SMN1; SMN2 (0.47) SMN1; SMN2NPC1RAB9ATSHRRECQL
SCHEMBL4865217 0.80 SMN1; SMN2 (0.55) SMN1; SMN2NPC1RAB9ACD274ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1047778-C Pyrimido [5-4-d] pyrimidines, drugs containing these compounds, their use and process for preparing them THOMAE GMBH DR K (DE) 1999-12-29 CN disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed