SCHEMBL8798945

SCHEMBL8798945

O=C1CN(S(=O)(=O)c2cc3c(Cl)c(Cl)ccc3o2)C(=S)N1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.31
PDE2A O00408 1/20 0.30
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
P2RY12 Q9H244 1/20 0.30
PKM P14618 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799930 0.89 MEN1 (0.35) MEN1KMT2APOLBTDP1PDE2A
SCHEMBL8799304 0.81 MEN1 (0.32) MEN1KMT2APOLBTDP1
SCHEMBL8798971 0.79 ALDH1A1 (0.32) POLB
SCHEMBL8799255 0.76 CA2 (0.46) MEN1KMT2APOLBL3MBTL1
SCHEMBL8798369 0.74 MEN1 (0.38) MEN1KMT2APOLBTDP1
SCHEMBL8789825 0.71 PKM (0.56) MEN1KMT2APOLBPKML3MBTL1
SCHEMBL8799859 0.71 MEN1 (0.34) MEN1KMT2APOLBTDP1PKM
SCHEMBL8799877 0.70 MEN1 (0.33) MEN1KMT2APOLBTDP1
SCHEMBL8799649 0.69 AHR (0.41) KMT2AL3MBTL1
SCHEMBL8800240 0.68 AKR1B1 (0.47) MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355827-B1 Hydantoin derivatives MOCHIDA PHARM CO LTD (JP) 1997-01-02 EP disclosed
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
WO-1990002126-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-03-08 WO disclosed
EP-0355827-A2 Hydantoin derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed