Veliflapon

Veliflapon

SCHEMBL8798993

O=C(O)[C@H](c1ccc(OCc2ccc3ccccc3n2)cc1)C1CCCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ALOX5AP

The experimentally established mechanism targets of Veliflapon. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 20/20 1.00
HDAC6 Q9UBN7 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Veliflapon SCHEMBL1004174 1.00 ALOX5 (1.00) ALOX5HDAC6
Veliflapon SCHEMBL29405516 1.00 ALOX5 (1.00) ALOX5HDAC6
Veliflapon SCHEMBL502932 1.00 ALOX5 (1.00) ALOX5HDAC6
Veliflapon SCHEMBL30386644 1.00 ALOX5 (1.00) ALOX5HDAC6
SCHEMBL2109295 0.99 ALOX5 (1.00) ALOX5HDAC6
SCHEMBL2110833 0.99 ALOX5 (1.00) ALOX5HDAC6
SCHEMBL7818529 0.99 ALOX5 (1.00) ALOX5HDAC6
SCHEMBL9123409 0.99 ALOX5 (1.00) ALOX5HDAC6
SCHEMBL9123415 0.99 ALOX5 (1.00) ALOX5HDAC6
SCHEMBL7818344 0.99 ALOX5 (1.00) ALOX5HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-8245593-A None JP disclosed
JP-8253448-A None JP disclosed
EP-0772594-A1 IMINOXYCARBOXYLATES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS Abbott Laboratories (US) 1997-05-14 EP disclosed
JP-H08253448-A HETEROCYCLIC SUBSTITUENT GROUP-CONTAINING OXY-PHENYL(PHENYL)GLYCINOL AMIDE BAYER AG 1996-10-01 JP disclosed
JP-H08245593-A 4-(QUINOLIN-2-YL-METHOXY)-PHENYL-ACETIC ACID DERIVATIVE BAYER AG 1996-09-24 JP disclosed
US-5512581-A ANTIINFLAMMATORY AGENT ABBOTT LABORATORIES (US) 1996-04-30 US disclosed
WO-1996002507-A1 IMINOXYCARBOXYLATES AND DERIVATIVES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1996-02-01 WO disclosed