SCHEMBL8799158

SCHEMBL8799158

N#Cc1ccc2sc(S(=O)(=O)N3CC(=O)NC3=O)cc2c1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 3/20 0.33
STS P08842 1/20 0.33
CA2 P00918 4/20 0.32
GAA P10253 1/20 0.31
G6PD P11413 1/20 0.31
CA1 P00915 1/20 0.31
FASN P49327 1/20 0.31
CLK1 P49759 1/20 0.31
DYRK1A Q13627 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
AKR1B1 P15121 1/20 0.31
CTSG P08311 1/20 0.30
MIF P14174 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797912 0.90 CMA1 (0.32) CMA1STSCA2GAA
SCHEMBL8799136 0.81 F10 (0.39) CMA1
SCHEMBL8798949 0.81 CA2 (0.34) CA2AKR1B1
SCHEMBL5953051 0.80 CA2 (0.49) CA2AKR1B1
SCHEMBL8797869 0.79 POLB (0.43) STSCA2
SCHEMBL8799290 0.74 F10 (0.47)
SCHEMBL8800196 0.73 TRPV4 (0.43) CA2CA1CLK1DYRK1ADYRK1B
SCHEMBL8799012 0.69 CA2 (0.46) CA2AKR1B1
SCHEMBL8799201 0.68 HDAC3 (0.37) CA2AKR1B1
SCHEMBL8799786 0.68 HDAC3 (0.37) CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355827-B1 Hydantoin derivatives MOCHIDA PHARM CO LTD (JP) 1997-01-02 EP disclosed
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
US-4914099-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-04-03 US disclosed
WO-1990002126-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-03-08 WO disclosed
EP-0355827-A2 Hydantoin derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed
WO-1989001934-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-09 WO disclosed
EP-0305947-A1 Hydantoin derivatives, process for their preparation and pharmaceutical compositions containing the same as well as their use MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-08 EP disclosed