SCHEMBL8799250

SCHEMBL8799250

O=C1NC(=O)C(S(=O)(=O)c2cccc3ccccc23)N1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
ALDH1A1 P00352 2/20 0.41
CASP1 P29466 1/20 0.41
AKR1B1 P15121 1/20 0.40
PRSS1 P07477 3/20 0.39
HTR6 P50406 3/20 0.39
F2 P00734 2/20 0.39
PRSS2 P07478 2/20 0.39
PRSS3 P35030 2/20 0.39
TSHR P16473 1/20 0.38
IDO1 P14902 1/20 0.37
C1R P00736 1/20 0.36
ATM Q13315 1/20 0.36
CNR1 P21554 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9784332 0.75 CA1 (0.44) CA1CA2CA9MEN1KMT2A
SCHEMBL8972696 0.74 MAPT (0.38) CA1CA2CA9ALDH1A1HTR6
SCHEMBL9000118 0.73 TSHR (0.47) CA1CA2CA9KMT2AALDH1A1
SCHEMBL6453126 0.72 KDM4E (0.49) CA1CA2CA9MEN1KMT2A
SCHEMBL20789878 0.68 CA1 (0.55) CA1CA2CA9MEN1KMT2A
SCHEMBL30588975 0.68 IDO1 (0.55) MEN1KMT2AALDH1A1CASP1AKR1B1
SCHEMBL10822158 0.68 IDO1 (0.55) MEN1KMT2AALDH1A1CASP1AKR1B1
SCHEMBL8966424 0.68 ALDH1A1 (0.54) MEN1KMT2AALDH1A1CASP1IDO1
SCHEMBL8547360 0.68 ALDH1A1 (0.54) MEN1KMT2AALDH1A1CASP1IDO1
SCHEMBL6113594 0.67 CA1 (0.63) CA1CA2CA9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0355827-B1 Hydantoin derivatives MOCHIDA PHARM CO LTD (JP) 1997-01-02 EP disclosed
EP-0444546-B1 Hydantoin derivatives for use as hypoglycemic and/or hypolipidemic agents MOCHIDA PHARM CO LTD (JP) 1996-09-11 EP disclosed
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
EP-0305947-B1 HYDANTOIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS WELL AS THEIR USE MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1992-07-29 EP disclosed
WO-1991012803-A1 HYDANTOIN DERIVATIVES FOR USE AS HYPOGLYCEMIC AND/OR HYPOLIPIDEMIC AGENTS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-09-05 WO disclosed
EP-0444546-A1 Hydantoin derivatives for use as hypoglycemic and/or hypolipidemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-09-04 EP disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
US-4914099-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-04-03 US disclosed
WO-1990002126-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-03-08 WO disclosed
EP-0355827-A2 Hydantoin derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-02-28 EP disclosed
WO-1989001934-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-09 WO disclosed