SCHEMBL8799607

SCHEMBL8799607

COc1cc(Cn2c(=O)c(OC(=O)O)c(-c3ccc4c(c3)OCO4)c3c(OC)c(OC)ccc32)cc(OC)c1OC

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 16/20 0.64
EDNRA P25101 9/20 0.51
ALDH1A1 P00352 2/20 0.43
MAPK1 P28482 1/20 0.43
KDM4E B2RXH2 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799661 0.92 EDNRB (0.61) EDNRBEDNRAALDH1A1MAPK1KDM4E
SCHEMBL8798950 0.89 EDNRB (0.81) EDNRBEDNRAALDH1A1MAPK1KDM4E
SCHEMBL8575962 0.89 EDNRB (0.81) EDNRBEDNRAALDH1A1MAPK1
SCHEMBL8798655 0.88 EDNRB (0.67) EDNRBEDNRAALDH1A1KDM4E
SCHEMBL8798300 0.87 EDNRB (0.71) EDNRBEDNRAALDH1A1KDM4E
SCHEMBL8578538 0.86 EDNRB (0.69) EDNRBEDNRAALDH1A1MAPK1KDM4E
SCHEMBL8799108 0.81 EDNRB (0.77) EDNRBEDNRAALDH1A1MAPK1KDM4E
SCHEMBL8798090 0.81 EDNRB (0.64) EDNRBEDNRAALDH1A1KDM4E
SCHEMBL8799772 0.80 EDNRB (0.68) EDNRBEDNRAALDH1A1KDM4E
SCHEMBL8576085 0.78 EDNRB (1.00) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0757039-A1 Endothelin receptor antagonists MERCK PATENT GmbH (DE) 1997-02-05 EP disclosed