SCHEMBL8799737

SCHEMBL8799737

CC(C)c1cc(Oc2c(Cl)cc(NC(=O)C(=O)OCc3ccccc3)cc2Cl)ccc1O

nearest known ligand 0.81

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
THRB P10828 9/20 0.59
THRA P10827 8/20 0.59
RORC P51449 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799735 0.85 THRA (0.67) THRBTHRA
SCHEMBL6903277 0.83 THRA (0.77) THRBTHRA
SCHEMBL9170838 0.82 RORC (0.47) THRBTHRARORC
SCHEMBL2043784 0.79 THRB (0.78) THRBTHRARORC
SCHEMBL2042956 0.78 THRB (0.69) THRBTHRARORC
SCHEMBL8798722 0.77 THRA (0.76) THRBTHRA
SCHEMBL4964368 0.77 THRB (0.63) THRBTHRARORC
SCHEMBL8894466 0.76 THRA (0.71) THRBTHRA
SCHEMBL29373235 0.74 THRA (1.00) THRBTHRA
SCHEMBL282382 0.74 THRA (1.00) THRBTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0580550-B1 Oxamic acid derivatives as hypocholesteremic agents CIBA GEIGY AG (CH) 1997-10-22 EP disclosed
US-5654468-A ANTILIPID, ANTICHOLESTEROL AGENTS CIBA-GEIGY CORPORATION (US) 1997-08-05 US disclosed
US-5569674-A ANTICHOLESTEROL AGENTS CIBA-GEIGY CORPORATION (US) 1996-10-29 US disclosed
US-5401772-A Anticholesterol agents with aromatic amines CIBA-GEIGY CORPORATION (US) 1995-03-28 US disclosed
EP-0580550-A1 Oxamic acid derivatives as hypocholesteremic agents CIBA-GEIGY AG (CH) 1994-01-26 EP disclosed