SCHEMBL8799883

SCHEMBL8799883

O=C1c2ccccc2C(=O)N1CCCc1cc2cc([N+](=O)[O-])ccc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.48
CYP19A1 P11511 2/20 0.48
GPR84 Q9NQS5 1/20 0.47
ALDH1A1 P00352 2/20 0.43
NR1H2 P55055 1/20 0.43
NR1H3 Q13133 1/20 0.43
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801068 0.81 GPR84 (0.51) GPR84ALDH1A1MEN1LMNAMAPT
SCHEMBL9486575 0.76 CYP19A1 (0.49) CYP19A1ALDH1A1MEN1LMNAMAPT
SCHEMBL8802605 0.76 CYP19A1 (0.49) CYP19A1ALDH1A1LMNAMAPT
SCHEMBL28923795 0.75 KCNH2 (0.50) CYP19A1ALDH1A1MEN1LMNAMAPT
SCHEMBL2125302 0.75 CYP19A1 (0.58) CYP19A1MEN1MAPTKMT2A
SCHEMBL10430003 0.75 CYP19A1 (0.48) CYP19A1ALDH1A1LMNAMAPT
SCHEMBL6620808 0.74 SIGMAR1 (0.60) ALDH1A1MEN1HTTKMT2A
SCHEMBL12758951 0.73 HRH3 (0.56) GPR84ALDH1A1MEN1LMNAMAPT
SCHEMBL6597520 0.73 CYP19A1 (0.51) CYP19A1ALDH1A1MEN1LMNAMAPT
SCHEMBL7807147 0.73 KDM4E (0.55) CYP19A1ALDH1A1MEN1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779887-A1 NOVEL BENZIMIDAZOLE DERIVATIVES HAVING CGMP-PHOSPHODISTERASE INHIBITING ACTIVITY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-06-25 EP disclosed