SCHEMBL8800166

SCHEMBL8800166

CC(=O)OC(C)c1nc(C(C)C)c(Sc2cc(F)cc(F)c2)n1Cc1cccnc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 3/20 0.37
GRIN2B Q13224 3/20 0.37
IDO1 P14902 2/20 0.35
S1PR3 Q99500 6/20 0.35
NOX4 Q9NPH5 2/20 0.33
RORC P51449 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
SRC P12931 1/20 0.33
GNRHR P30968 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974251 0.93 GRIN1 (0.38) GRIN1GRIN2BIDO1S1PR3
SCHEMBL6974146 0.90 ALDH1A1 (0.36) S1PR3NOX4
SCHEMBL8800346 0.89 MEN1 (0.32) GNRHR
SCHEMBL8801330 0.89 KDM4E (0.38) S1PR3NOX4
SCHEMBL8801745 0.86 ALDH1A1 (0.40) GRIN1GRIN2B
SCHEMBL6969897 0.86 GRIN1 (0.38) GRIN1GRIN2BIDO1S1PR3NOX4
SCHEMBL7079752 0.84 GRIN1 (0.37) GRIN1GRIN2BIDO1S1PR3NOX4
SCHEMBL7080221 0.83 GNRHR (0.37) GNRHR
SCHEMBL8799639 0.83 GRIN1 (0.35) GRIN1GRIN2B
SCHEMBL6961698 0.83 S1PR3 (0.38) S1PR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed