SCHEMBL8801745

SCHEMBL8801745

CC(=O)OC(C)c1nc(C(C)C)c(Sc2cccc(Cl)c2)n1Cc1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
TP53 P04637 3/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
GABRA5 P31644 2/20 0.34
NPC1 O15118 2/20 0.34
GABRA1 P14867 1/20 0.34
P2RX7 Q99572 1/20 0.34
PKM P14618 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
KMT2A Q03164 1/20 0.34
PTGER2 P43116 1/20 0.34
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974146 0.93 ALDH1A1 (0.36) ALDH1A1TP53TDP1GABRA5GABRA1
SCHEMBL8801551 0.91 TDP1 (0.36) ALDH1A1LMNATP53TDP1KMT2A
SCHEMBL6974251 0.90 GRIN1 (0.38) ALDH1A1LMNAGRIN1GRIN2BPKM
SCHEMBL8801330 0.89 KDM4E (0.38) ALDH1A1LMNA
SCHEMBL7080221 0.87 GNRHR (0.37) ALDH1A1LMNAKMT2A
SCHEMBL6971953 0.86 ALDH1A1 (0.41) ALDH1A1LMNATP53GRIN1GRIN2B
SCHEMBL8800166 0.86 GRIN1 (0.37) GRIN1GRIN2B
SCHEMBL6967425 0.85 ALDH1A1 (0.40) ALDH1A1LMNATP53GRIN1GRIN2B
SCHEMBL8802789 0.85 TP53 (0.37) ALDH1A1LMNATP53TDP1NPC1
SCHEMBL7086183 0.84 TP53 (0.35) ALDH1A1TP53GRIN1GRIN2BTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed