SCHEMBL6961698

SCHEMBL6961698

CC(=O)OC(C)c1nc(C(C)C)c(Sc2cc(F)cc(F)c2)n1Cc1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 17/20 0.38
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
GFER P55789 1/20 0.33
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799402 0.93 S1PR3 (0.37) S1PR3ALDH1A1SYK
SCHEMBL8800780 0.90 PTGDR2 (0.35) ALDH1A1KDM4E
SCHEMBL8800407 0.89 MEN1 (0.33) S1PR3ALDH1A1KDM4E
SCHEMBL7086183 0.86 TP53 (0.35) ALDH1A1KDM4E
SCHEMBL7082930 0.85 S1PR3 (0.38) S1PR3ALDH1A1KDM4ELMNAGFER
SCHEMBL8800346 0.84 MEN1 (0.32) LMNA
SCHEMBL6973461 0.84 S1PR3 (0.39) S1PR3ALDH1A1KDM4ELMNAGFER
SCHEMBL8800166 0.83 GRIN1 (0.37) S1PR3
SCHEMBL8800655 0.83 CFTR (0.41) S1PR3ALDH1A1KDM4ELMNA
SCHEMBL6974419 0.83 ALDH1A1 (0.31) ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed