SCHEMBL8800296

SCHEMBL8800296

CC(=O)c1ccc(OC(C)C)c([N+](=O)[O-])c1

nearest known ligand 0.72

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.72
POLB P06746 6/20 0.53
ALDH1A1 P00352 6/20 0.51
KMT2A Q03164 4/20 0.51
LMNA P02545 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
HPGD P15428 1/20 0.51
TSHR P16473 2/20 0.48
CYP3A4 P08684 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MAPT P10636 4/20 0.48
XDH P47989 1/20 0.47
MEN1 O00255 3/20 0.46
RECQL P46063 1/20 0.46
PKM P14618 1/20 0.46
PDE7A Q13946 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16956345 0.89 PDK1 (0.70) PDK1POLBALDH1A1KMT2ALMNA
SCHEMBL2550259 0.88 PDK1 (0.72) PDK1ALDH1A1KMT2ALMNAHPGD
SCHEMBL6112853 0.87 PDK1 (0.71) PDK1POLBALDH1A1KMT2ALMNA
SCHEMBL28748723 0.87 PDK1 (0.75) PDK1POLBALDH1A1KMT2ALMNA
SCHEMBL28317018 0.85 PDK1 (0.69) PDK1POLBALDH1A1KMT2ALMNA
SCHEMBL31439475 0.85 PDK1 (0.69) PDK1POLBALDH1A1KMT2ALMNA
SCHEMBL6113956 0.85 PDK1 (0.69) PDK1POLBALDH1A1KMT2ALMNA
SCHEMBL31397869 0.84 PDK1 (0.85) PDK1POLBALDH1A1KMT2ALMNA
SCHEMBL31397863 0.84 PDK1 (0.76) PDK1POLBALDH1A1KMT2ALMNA
SCHEMBL5913273 0.84 PDK1 (0.67) PDK1POLBALDH1A1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119977942-A Quinazolinone derivative for inducing iron death as well as synthesis method and application thereof 西安交通大学 2025-05-13 CN disclosed
WO-2025015167-A2 ERASTIN KETONE ANALOGS AND USES THEREOF EXARTA THERAPEUTICS, INC. (US) 2025-01-16 WO disclosed
US-9938245-B2 Carbonyl erastin analogs and their use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-04-10 US disclosed
US-9938245-B2 Carbonyl erastin analogs and their use THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2018-04-10 US disclosed
US-20160332974-A1 CARBONYL ERASTIN ANALOGS AND THEIR USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2016-11-17 US disclosed
US-20160332974-A1 CARBONYL ERASTIN ANALOGS AND THEIR USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2016-11-17 US disclosed
WO-2015109009-A1 CARBONYL ERASTIN ANALOGS AND THEIR USE THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-07-23 WO disclosed
EP-0482771-B1 Heterocyclic acids ZENECA LTD (GB) 1997-06-18 EP disclosed
US-5219874-A Heterocyclic acids IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-06-15 US disclosed
EP-0482771-A2 Heterocyclic acids ZENECA LIMITED (GB) 1992-04-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160332974-A1 CARBONYL ERASTIN ANALOGS AND THEIR USE KEAP1, GPX1, GPX4 PDK1 673/4885POLB 4261/4885ALDH1A1 407/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.