SCHEMBL8800567

SCHEMBL8800567

CC(C)[C@H](NC(=O)CC1OC1C(Cc1ccccc1)NC(=O)[C@H](NC(=O)c1ccc2ccccc2n1)C(C)C)C(=O)NCc1ccccn1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSD P07339 4/20 0.61
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TSHR P16473 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
CYP3A4 P08684 1/20 0.42
REN P00797 2/20 0.41
CTSE P14091 1/20 0.41
CA2 P00918 1/20 0.40
HDAC1 Q13547 1/20 0.39
CCR1 P32246 1/20 0.39
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8800938 0.92 CTSD (0.74) CTSDALDH1A1SMN1; SMN2TSHRCYP1A2
SCHEMBL8801074 0.88 CTSD (0.69) CTSDALDH1A1MAPTRENHDAC1
SCHEMBL8801445 0.86 CTSD (0.70) CTSDALDH1A1SMN1; SMN2TSHRCYP1A2
SCHEMBL8800743 0.86 CTSD (0.59) CTSDALDH1A1SMN1; SMN2TSHRCYP1A2
SCHEMBL8801114 0.86 CTSD (0.66) CTSDALDH1A1RENHDAC1CCR1
SCHEMBL7299644 0.83 CTSD (0.62) CTSDALDH1A1SMN1; SMN2MAPTHDAC1
SCHEMBL8800871 0.79 CTSD (0.86) CTSDALDH1A1CYP2D6CYP3A4REN
SCHEMBL8800288 0.79 CTSD (0.73) CTSDALDH1A1CYP1A2CYP2D6MAPT
SCHEMBL8802750 0.78 CTSD (0.76) CTSDALDH1A1CYP2D6CYP3A4REN
SCHEMBL8801929 0.77 CTSD (0.82) CTSDALDH1A1CYP2D6CYP3A4REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP claimed
EP-0601486-A1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD. (KR) 1994-06-15 EP claimed