SCHEMBL8801074

SCHEMBL8801074

CC(C)[C@H](NC(=O)CC1OC1C(Cc1ccccc1)NC(=O)[C@H](NC(=O)c1ccc2ccccc2n1)C(C)C)C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSD P07339 4/20 0.69
CCR1 P32246 1/20 0.44
REN P00797 2/20 0.39
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
HDAC1 Q13547 2/20 0.38
CTSK P43235 3/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
PSMB5 P28074 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801114 0.93 CTSD (0.66) CTSDCCR1RENOPRM1OPRK1
SCHEMBL8800871 0.90 CTSD (0.86) CTSDCCR1RENOPRM1OPRK1
SCHEMBL7299644 0.90 CTSD (0.62) CTSDCCR1OPRM1OPRK1TMEM97
SCHEMBL8800567 0.88 CTSD (0.61) CTSDCCR1RENHDAC1ALDH1A1
SCHEMBL8800743 0.87 CTSD (0.59) CTSDCCR1RENHDAC1PSMB5
SCHEMBL8801929 0.83 CTSD (0.82) CTSDCCR1RENOPRM1OPRK1
SCHEMBL7313674 0.83 CTSD (0.80) CTSDCCR1RENOPRM1OPRK1
SCHEMBL8800938 0.80 CTSD (0.74) CTSDRENOPRM1OPRK1HDAC1
SCHEMBL8800288 0.79 CTSD (0.73) CTSDCCR1RENOPRM1OPRK1
SCHEMBL8801937 0.79 CTSD (0.78) CTSDCCR1RENOPRM1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601486-B1 Cis-epoxide derivatives useful as irreversible HIV protease inhibitors and process and intermediates for their preparation LUCKY LTD (KR) 1997-10-29 EP claimed