SCHEMBL8800748

SCHEMBL8800748

O=C(C(=O)c1ccccc1-c1ccccc1Cl)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 9/20 0.55
CES1 P23141 8/20 0.55
ALDH1A1 P00352 2/20 0.48
SMO Q99835 1/20 0.44
CYP2A6 P11509 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
HPGD P15428 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MAPK14 Q16539 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29972427 0.88 CES2 (0.67) CES2CES1ALDH1A1RAB9ATSHR
SCHEMBL24043882 0.85 CES2 (0.53) CES2CES1ALDH1A1HSP90AA1NPC1
SCHEMBL29468149 0.84 CES2 (0.78) CES2CES1ALDH1A1SMONPC1
SCHEMBL2225523 0.84 CES2 (0.78) CES2CES1ALDH1A1SMONPC1
SCHEMBL27803960 0.83 AKR1C3 (0.53) CES2CES1ALDH1A1SMOGAA
SCHEMBL2930892 0.80 ALDH1A1 (0.68) CES2CES1ALDH1A1CYP2A6GAA
Urea SCHEMBL28476564 0.79 CES2 (0.69) CES2CES1ALDH1A1SMONPC1
SCHEMBL5076702 0.79 TSHR (0.62) CES2CES1ALDH1A1SMOTSHR
SCHEMBL2141156 0.79 CES2 (0.54) CES2CES1ALDH1A1HSP90AA1HPGD
SCHEMBL8802307 0.79 CES2 (0.39) CES2CES1ALDH1A1SMOPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772601-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-05-14 EP disclosed
CN-86107695-A The 3-piperidine carboxylic acid of different nitrogen-replacements or the 3-pyridine carboxylic acid of nitrogen-replacement and their derivative 1987-05-13 CN disclosed