SCHEMBL8801165

SCHEMBL8801165

CCCCCCc1ccc(CN(C(N)=Nc2ccccc2)c2ccc(CCCCCC)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 3/20 0.47
HTR2A P28223 2/20 0.43
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
KCNH2 Q12809 1/20 0.42
SIGMAR1 Q99720 2/20 0.41
ESR1 P03372 2/20 0.41
ADRA2A P08913 2/20 0.41
ADORA3 P0DMS8 2/20 0.41
TACR2 P21452 2/20 0.41
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
SHBG P04278 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4977836 0.89 STAT3 (0.41) STAT3HTR2AITGB1ITGA4CYP3A4
SCHEMBL4984243 0.78 NR1H4 (0.42) KDM4ELTB4R2
SCHEMBL4982720 0.78 CYP3A4 (0.46) CYP3A4CYP2D6CYP2C9ADRA2AADRA2B
SCHEMBL8802180 0.77 ESR1 (0.49) STAT3HTR2ACYP3A4ESR1ADRA2A
SCHEMBL28751547 0.73 CNR2 (0.51) STAT3HTR2ACYP3A4ESR1ADRA2A
SCHEMBL8801161 0.72 STAT3 (0.47) STAT3KCNH2CNR2
SCHEMBL28887265 0.72 STAT3 (0.53) STAT3CNR2
SCHEMBL3921499 0.72 SIGMAR1 (0.51) SIGMAR1ADRA2AALDH1A1TP53ADRA2B
SCHEMBL3919033 0.72 MEN1 (0.54) SIGMAR1ADRA2AALDH1A1TP53ADRA2B
SCHEMBL855620 0.72 HDAC6 (0.55) STAT3ALDH1A1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0751767-A4 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE INC (US) 1997-12-10 EP claimed
EP-0751767-A1 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1997-01-08 EP claimed
WO-1995020950-A1 THERAPEUTIC GUANIDINES CAMBRIDGE NEUROSCIENCE, INC. (US) 1995-08-10 WO claimed