SCHEMBL8801570

SCHEMBL8801570

O=C(O)Oc1cn(-c2ccc(Cn3ccnn3)cc2)c2c(Cl)c(F)c(F)cc2c1=O

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 3/20 0.37
CYP19A1 P11511 5/20 0.36
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
HSP90AA1 P07900 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
STAT3 P40763 1/20 0.32
HSD17B1 P14061 2/20 0.31
HSD17B2 P37059 2/20 0.31
CHRM1 P11229 1/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2C9 P11712 2/20 0.31
MAPK8 P45983 1/20 0.31
KLKB1 P03952 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803908 0.94 ALDH1A1 (0.40) PIM1CYP19A1KDM4EALDH1A1POLB
SCHEMBL8801565 0.89 PIM1 (0.47) PIM1CYP19A1KDM4EALDH1A1POLB
SCHEMBL8802774 0.86 CYP3A4 (0.36) PIM1CYP19A1KDM4EALDH1A1POLB
SCHEMBL8801865 0.86 CYP19A1 (0.38) CYP19A1KDM4EALDH1A1IDO1TDO2
SCHEMBL8801306 0.85 PIM1 (0.37) PIM1CYP19A1KDM4EALDH1A1POLB
SCHEMBL8802022 0.84 CYP3A4 (0.35) CYP19A1KDM4EALDH1A1POLBHSP90AA1
SCHEMBL8801505 0.84 HPGD (0.42) CYP19A1KDM4EALDH1A1POLBHSP90AA1
SCHEMBL8803705 0.84 HDAC1 (0.38) PIM1CYP19A1KDM4EALDH1A1POLB
SCHEMBL8803902 0.82 ALDH1A1 (0.52) PIM1CYP19A1KDM4EALDH1A1POLB
SCHEMBL9048087 0.81 KDM4E (0.41) PIM1KDM4EALDH1A1POLBHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612731-B1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1997-08-20 EP disclosed
EP-0612731-A1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1994-08-31 EP disclosed