SCHEMBL8801892

SCHEMBL8801892

O=Cc1ccnc(-c2ccc(F)cc2F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 3/20 0.49
KDM1A O60341 6/20 0.45
HDAC1 Q13547 3/20 0.45
HDAC6 Q9UBN7 3/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC5 Q9UQL6 1/20 0.42
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
FAAH O00519 1/20 0.38
ALPL P05186 2/20 0.38
KDM4A O75164 1/20 0.36
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4938913 0.81 KDM1A (0.51) KDM1AHDAC1HDAC6HDAC2HDAC11
SCHEMBL29445848 0.81 KMO (0.54) KMOKDM1AMEN1KMT2AFAAH
SCHEMBL19072696 0.81 KMO (0.54) KMOKDM1AMEN1KMT2AFAAH
SCHEMBL8802396 0.80 KMO (0.46) KMOKDM1AHDAC1HDAC6HDAC2
SCHEMBL9939619 0.78 MEN1 (0.44) KDM1AHDAC1HDAC6HDAC5MEN1
SCHEMBL9607471 0.77 ALDH1A1 (0.45) KMOHDAC1HDAC6HDAC2HDAC11
SCHEMBL14879562 0.77 ALDH1A1 (0.49) MEN1KMT2AALDH1A1POLBHPGD
SCHEMBL730405 0.76 CCR1 (0.42) ALDH1A1KDM4AKDM4CRAB9A
SCHEMBL29387096 0.76 CCR1 (0.42) ALDH1A1KDM4AKDM4CRAB9A
SCHEMBL19847066 0.76 KDM1A (0.40) KDM1AHDAC1HDAC6HDAC2HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0695751-B1 AGENT ACTING ON THE CENTRAL NERVOUS SYSTEM, PROCESS FOR ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT VITA INVEST SA (ES) 1997-03-26 EP disclosed
EP-0695751-A1 AGENT ACTING ON THE CENTRAL NERVOUS SYSTEM, PROCESS FOR ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT VITA-INVEST, S.A. (ES) 1996-02-07 EP disclosed