SCHEMBL8802153

SCHEMBL8802153

NC1=NSNc2nc(-c3ccccc3)cnc21

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ATR Q13535 11/20 0.46
TLR9 Q9NR96 1/20 0.40
NOS1 P29475 1/20 0.39
PRKDC P78527 2/20 0.38
MAPK1 P28482 1/20 0.38
GSK3B P49841 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8802152 0.88 ATR (0.49) ATRTLR9NOS1PRKDCGSK3B
SCHEMBL8802240 0.73 XDH (0.37)
SCHEMBL8800858 0.71 ATR (0.41) ATRTLR9NOS1PRKDCMAPK1
SCHEMBL6701248 0.69 ATR (0.66) ATRTLR9PRKDC
SCHEMBL32688927 0.69 ATR (0.66) ATRTLR9PRKDC
SCHEMBL29519952 0.68 ATR (0.56) ATRTLR9NOS1PRKDCMAPK1
SCHEMBL12489014 0.68 ATR (0.56) ATRTLR9NOS1PRKDCMAPK1
SCHEMBL8800693 0.67 ATR (0.38) ATRTLR9NOS1MAPK1NPC1
SCHEMBL87574 0.66 CKS1B (0.55) ATRTLR9MAPK1NPC1RAB9A
SCHEMBL29406280 0.64 CKS1B (0.53) ATRTLR9MAPK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0580916-B1 N(1) substituted pyrazino [2,3-c]-1,2,6-thiadiazine 2,2-dioxides and their use as pharmaceuticals PRODESFARMA SA (ES) 1997-03-05 EP claimed