SCHEMBL8804203

SCHEMBL8804203

N#Cc1c(O)c2cccnc2n(-c2ccccc2)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.54
PDE4A P27815 7/20 0.50
PDE4B Q07343 6/20 0.50
PDE4C Q08493 6/20 0.50
PDE4D Q08499 6/20 0.50
ALDH1A1 P00352 3/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
PDE1A P54750 1/20 0.46
PDE1B Q01064 1/20 0.46
LOXL3 P58215 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
CACNA1B Q00975 1/20 0.42
APBA1 Q02410 1/20 0.42
LDHA P00338 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9715610 0.80 FEN1 (0.58) FEN1PDE4APDE4BPDE4CPDE4D
SCHEMBL10412161 0.80 FEN1 (0.58) FEN1PDE4APDE4BPDE4CPDE4D
SCHEMBL28978594 0.80 MAT2A (0.50) ALDH1A1TSHRMEN1KMT2AKDM4E
SCHEMBL29417532 0.80 MAT2A (0.50) ALDH1A1TSHRMEN1KMT2AKDM4E
SCHEMBL30084688 0.77 PIK3CG (0.40) FEN1PDE4APDE4BPDE4CPDE4D
SCHEMBL10421586 0.77 FEN1 (0.56) FEN1PDE4APDE4BPDE4CPDE4D
SCHEMBL29417554 0.77 ALDH1A1 (0.37) ALDH1A1TSHRMEN1KMT2AKDM4E
SCHEMBL28978832 0.77 MAT2A (0.42) ALDH1A1MEN1KMT2AGAA
SCHEMBL28978823 0.77 ALDH1A1 (0.37) ALDH1A1TSHRMEN1KMT2AKDM4E
SCHEMBL29417557 0.77 MAT2A (0.42) ALDH1A1MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526840-B1 Condensed naphthyridine derivatives KYOWA HAKKO KOGYO KK (JP) 1997-10-22 EP disclosed
US-5281610-A Pyrazolonaphthyridine pharmaceuticals KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-01-25 US disclosed
EP-0526840-A1 Condensed naphthyridine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-02-10 EP disclosed