SCHEMBL8804591

SCHEMBL8804591

CC(C)c1ccc(CN2CCN(C(c3ccc(F)cc3)c3ccc(F)cc3)CC2C)c(=O)c(N(C)CCN(C)C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 11/20 0.38
TACR1 P25103 3/20 0.33
ACHE P22303 2/20 0.32
LMNA P02545 1/20 0.32
CHRM2 P08172 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CHRM1 P11229 1/20 0.32
DRD2 P14416 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
CNR1 P21554 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
ADRA1A P35348 1/20 0.32
HRH1 P35367 1/20 0.32
OPRM1 P35372 1/20 0.32
DRD3 P35462 1/20 0.32
OPRK1 P41145 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448064 0.88 SLC6A3 (0.34) TACR1ACHELMNACHRM2ADORA3
SCHEMBL7437175 0.85 ACHE (0.46) ACHELMNACHRM2ADORA3CHRM1
SCHEMBL7434590 0.82 ACHE (0.43) ACHELMNACHRM2ADORA3CHRM1
SCHEMBL7436646 0.81 LMNA (0.45) SLC6A9TACR1ACHELMNACHRM2
SCHEMBL7444396 0.78 ACHE (0.46) ACHELMNACHRM2ADORA3CHRM1
SCHEMBL7442593 0.77 MEN1 (0.43) LMNACHRM2ADORA3CHRM1DRD2
SCHEMBL7436788 0.76 ACHE (0.44) ACHELMNACHRM2ADORA3CHRM1
SCHEMBL7496645 0.73 MEN1 (0.44) ACHELMNACHRM2ADORA3CHRM1
SCHEMBL7447472 0.73 HRH1 (0.48) SLC6A9LMNACHRM2ADORA3CHRM1
SCHEMBL8805485 0.73 CACNA2D1 (0.42) LMNAADORA3CNR1HRH1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0546102-B1 TROPOLONE DERIVATIVES AND PHARMACEUTICAL COMPOSITION THEREOF FOR PREVENTING AND TREATING ISCHEMIC DISEASES UPJOHN CO (US) 1997-10-15 EP claimed
US-5594144-A TREATING CEREBROVASCULAR AND CARDIOVASCULAR DISORDERS THE UPJOHN COMPANY (US) 1997-01-14 US disclosed