SCHEMBL8804625

SCHEMBL8804625

COc1cc(CNC(C)C(N)=O)cc(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.53
MAOB P27338 4/20 0.50
SCN9A Q15858 2/20 0.48
TACR1 P25103 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803423 0.90 MAOA (0.48) MAOAMAOBSCN9A
SCHEMBL8803242 0.85 MAOB (0.64) MAOAMAOBSCN9AMEN1KMT2A
SCHEMBL9201087 0.84 MAOA (0.62) MAOAMAOBSCN9A
SCHEMBL8804579 0.84 MAOA (0.62) MAOAMAOBSCN9A
Hydrochloric Acid SCHEMBL5967428 0.83 MAOA (0.61) MAOAMAOBSCN9A
SCHEMBL17666275 0.80 MAOA (0.65) MAOAMAOBSCN9A
SCHEMBL23440934 0.79 MAOB (0.65) MAOAMAOBSCN9A
SCHEMBL8802147 0.78 ALDH1A1 (0.60) MAOAMAOBSCN9AMEN1KMT2A
SCHEMBL21346322 0.77 TSHR (0.53) TACR1MEN1KMT2A
SCHEMBL23440921 0.77 MAOB (0.67) MAOAMAOBSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775140-A1 SPIRO-SUBSTITUTED AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1997-05-28 EP disclosed
WO-1996005203-A1 SPIRO-SUBSTITUTED AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1996-02-22 WO disclosed