SCHEMBL8804579

SCHEMBL8804579

COc1ccc(CNC(C)C(N)=O)cc1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.62
SCN9A Q15858 2/20 0.59
MAOB P27338 3/20 0.57
HRH3 Q9Y5N1 3/20 0.56
HRH1 P35367 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9201087 1.00 MAOA (0.62) MAOASCN9AMAOBHRH3HRH1
Hydrochloric Acid SCHEMBL5967428 0.98 MAOA (0.61) MAOASCN9AMAOBHRH3HRH1
SCHEMBL17666275 0.95 MAOA (0.65) MAOASCN9AMAOBHRH3HRH1
SCHEMBL23440921 0.92 MAOB (0.67) MAOASCN9AMAOBHRH3HRH1
SCHEMBL28424984 0.90 MAOA (0.60) MAOASCN9AMAOBHRH3HRH1
SCHEMBL2716941 0.89 ALDH1A1 (0.51) MAOA
SCHEMBL6237220 0.85 LDHA (0.57)
SCHEMBL28049334 0.85 LDHA (0.57)
SCHEMBL14971737 0.85 ALDH1A1 (0.51) MAOA
SCHEMBL8804625 0.84 MAOA (0.53) MAOASCN9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775140-A1 SPIRO-SUBSTITUTED AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1997-05-28 EP claimed
WO-1996005203-A1 SPIRO-SUBSTITUTED AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1996-02-22 WO claimed
EP-0680469-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1995-11-08 EP disclosed
WO-1994017035-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME DR. KARL THOMAE GMBH (DE) 1994-08-04 WO disclosed