SCHEMBL8807992

SCHEMBL8807992

CS(=O)(=O)OCCC1(c2ccc3ccccc3c2)CC(=O)N(Cc2ccccc2)C1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.41
TACR1 P25103 16/20 0.40
TACR2 P21452 2/20 0.38
TACR3 P29371 2/20 0.38
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8347511 0.82 KDM4E (0.45) CCR5TACR1TACR2TACR3KDM4E
SCHEMBL8808253 0.81 CCR5 (0.44) CCR5TACR1TACR2TACR3KDM4E
SCHEMBL8296291 0.78 TACR1 (0.63) TACR1TACR2TACR3
SCHEMBL8366723 0.78 TACR1 (0.49) TACR1TACR2TACR3
SCHEMBL7765748 0.76 CCR5 (0.41) CCR5TACR1TACR2TACR3
SCHEMBL7947464 0.74 CCR5 (0.54) CCR5TACR1TACR2TACR3
SCHEMBL4631694 0.74 TACR1 (0.46) TACR1TACR2TACR3
SCHEMBL7847578 0.73 TACR1 (0.61) CCR5TACR1TACR2TACR3
SCHEMBL8355624 0.71 TACR1 (0.52) CCR5TACR1TACR2TACR3
SCHEMBL8884449 0.71 TACR2 (0.55) TACR1TACR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696280-B1 SUBSTITUTED PYRROLIDIN-3-YL-ALKYL-PIPERIDINES USEFUL AS TACHYKININ ANTAGONISTS MERRELL PHARMA INC (US) 1997-09-24 EP disclosed