SCHEMBL8808680

SCHEMBL8808680

CCOc1nncc2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.52
POLB P06746 3/20 0.52
ALDH1A1 P00352 4/20 0.50
MAPK1 P28482 1/20 0.49
CYP1A2 P05177 2/20 0.47
CYP2D6 P10635 2/20 0.47
HIF1A Q16665 1/20 0.47
HTT P42858 1/20 0.46
TDP1 Q9NUW8 2/20 0.46
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
TP53 P04637 4/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
MAPT P10636 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 2/20 0.43
CYP3A4 P08684 2/20 0.43
GOT1 P17174 2/20 0.43
MPO P05164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2488955 0.98 LMNA (0.51) LMNAPOLBALDH1A1MAPK1CYP1A2
SCHEMBL8811067 0.86 ALDH1A1 (0.48) LMNAPOLBALDH1A1MAPK1CYP1A2
SCHEMBL8809641 0.79 ALDH1A1 (0.59) LMNAPOLBALDH1A1MAPK1CYP1A2
SCHEMBL29674926 0.79 ALDH1A1 (0.59) LMNAPOLBALDH1A1MAPK1CYP1A2
SCHEMBL9461493 0.79 LMNA (0.56) LMNAPOLBALDH1A1MAPK1CYP1A2
SCHEMBL16115497 0.78 ALDH1A1 (0.56) LMNAPOLBALDH1A1CYP1A2HTT
SCHEMBL599375 0.77 LMNA (0.51) LMNAPOLBALDH1A1MAPK1CYP1A2
SCHEMBL8129269 0.76 CYP1A2 (0.42) LMNAPOLBALDH1A1MAPK1CYP1A2
SCHEMBL30418421 0.76 CYP1A2 (0.42) LMNAPOLBALDH1A1MAPK1CYP1A2
SCHEMBL21965729 0.75 LMNA (0.43) LMNAPOLBALDH1A1MAPK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0539805-B1 Phthalazines substituted on position 1 by an ether group and process for their preparation ASTA MEDICA AG (DE) 1997-09-03 EP claimed
US-5354750-A Analgesics, antinflammatory, anticonvulsive and antipyretic agents ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1994-10-11 US claimed
EP-0539805-A1 Phthalazines substituted on position 1 by an ether or a thioether group and process for their preparation ASTA Medica Aktiengesellschaft (DE) 1993-05-05 EP claimed
JP-5222002-A None JP disclosed
EP-0539805-B1 Phthalazines substituted on position 1 by an ether group and process for their preparation ASTA MEDICA AG (DE) 1997-09-03 EP disclosed
US-5354750-A Analgesics, antinflammatory, anticonvulsive and antipyretic agents ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1994-10-11 US disclosed
JP-H05222002-A PHTHALAZINE CONTAINING ETHER OR THIOETHER GROUP IN 1-POSITION, ITS PREPARATION AND PHARMACEUTICAL CONTAINING THE SAME, WHICH HAS ANALGESIC, ANTI-INFLAMMATORY, ANTICONVULSIVE AND ANTI-PYRETIC ACTION, AND THEIR PREPARATION ASTA MEDICA AG 1993-08-31 JP disclosed
EP-0539805-A1 Phthalazines substituted on position 1 by an ether or a thioether group and process for their preparation ASTA Medica Aktiengesellschaft (DE) 1993-05-05 EP disclosed
US-5037719-A Image forming method using microcapsules containing silver halide and a salt of a reducing agent FUJI PHOTO FILM CO., LTD. (JP) 1991-08-06 US disclosed
US-4970132-A CLARITY OF IMAGE; STORAGE STABILITY FUJI PHOTO FILM CO., LTD. (JP) 1990-11-13 US disclosed
US-4902599-A CONTAINING HYDRAZIDE AND HYDROZINE COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 1990-02-20 US disclosed
EP-0219087-A2 Light-sensitive material FUJI PHOTO FILM CO., LTD. (JP) 1987-04-22 EP disclosed