SCHEMBL8808909

SCHEMBL8808909

COc1ccc2c(c1)c(OCC(=O)Nc1cccnc1)nn2Cc1ccc(Cl)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.55
NOTUM Q6P988 4/20 0.50
PDE4A P27815 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
KCNH2 Q12809 2/20 0.47
PDE6D O43924 1/20 0.46
TP53 P04637 1/20 0.46
NPC1 O15118 2/20 0.46
ATM Q13315 1/20 0.46
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
RAB9A P51151 1/20 0.45
LMNA P02545 3/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8813770 0.92 NOTUM (0.49) PTGS2NOTUMKCNH2PDE6DNPC1
SCHEMBL8810241 0.90 LMNA (0.52) PTGS2KCNH2NPC1ALDH1A1RAB9A
SCHEMBL8807554 0.87 NOTUM (0.53) NOTUMKCNH2NPC1ATMALDH1A1
SCHEMBL8812598 0.82 MEN1 (0.50) PTGS2TP53KDM4ECYP1A2CYP3A4
SCHEMBL8806408 0.79 KCNH2 (0.52) KCNH2TP53ALDH1A1KDM4ECYP1A2
SCHEMBL8808912 0.79 NOTUM (0.54) NOTUMKCNH2NPC1ALDH1A1KDM4E
SCHEMBL8811999 0.76 YES1 (0.54) TP53NPC1RAB9ALMNAMAPK1
SCHEMBL9058581 0.75 HTT (0.43) TP53NPC1ATMKDM4ERAB9A
SCHEMBL2168483 0.74 PDE4A (0.57) PTGS2PDE4APDE4BPDE4CPDE4D
SCHEMBL2999650 0.74 PDE4A (0.64) PTGS2PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775131-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA Medica Aktiengesellschaft (DE) 1997-05-28 EP disclosed
WO-1996004266-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1996-02-15 WO disclosed