SCHEMBL8809126

SCHEMBL8809126

CC1(C)CCC(C)(C)c2cc3c(cc21)SCCC3=O

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 1/20 0.53
HTT P42858 1/20 0.50
VHL P40337 1/20 0.46
ELOC Q15369 1/20 0.46
ELOB Q15370 1/20 0.46
RXRA P19793 8/20 0.35
RARA P10276 6/20 0.35
CYP26B1 Q9NR63 4/20 0.35
RXRG P48443 3/20 0.35
CYP26A1 O43174 3/20 0.35
CA2 P00918 2/20 0.33
RARB P10826 6/20 0.33
RXRB P28702 2/20 0.33
CYP3A4 P08684 1/20 0.32
RARG P13631 5/20 0.31
RYR2 Q92736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809982 0.78 HIF1A (0.41) RXRARARACYP26B1RXRGCYP26A1
SCHEMBL8310387 0.73 RXRA (0.36) RXRARARACYP26B1RXRGCYP26A1
SCHEMBL7624438 0.72 PBRM1 (0.44) RXRARARARXRGRARBRXRB
SCHEMBL2194526 0.70 MAOB (0.46) ALDH1A1RXRARARARXRG
SCHEMBL9607758 0.69 KDM4E (0.56) KDM4EALDH1A1HTTVHLELOC
SCHEMBL10363739 0.69 KDM4E (0.56) KDM4EALDH1A1HTTVHLELOC
SCHEMBL10364205 0.69 VHL (0.62) KDM4EALDH1A1HTTVHLELOC
SCHEMBL6915238 0.69 MEN1 (0.51)
SCHEMBL8471642 0.69 KDM4E (1.00) KDM4EALDH1A1HTTVHLELOC
SCHEMBL10890090 0.68 KDM4E (0.54) KDM4EALDH1A1HTTVHLELOC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1173497-A Heterocycle-containing carbonic acid derivatives EISAI CO LTD (JP) 1998-02-18 CN disclosed
EP-0638071-B1 HETEROCYCLIC CARBONIC ACID DERIVATIVES WHICH BIND TO RETINOID RECEPTORS (RAR) EISAI CO LTD (JP) 1997-04-09 EP disclosed
US-5612356-A RETINOID ANTAGONISTS EISAI CO., LTD. (JP) 1997-03-18 US disclosed
CN-1094052-A Heterocyclic ring-containing carbonic acid derivatives EISAI CO LTD (JP) 1994-10-26 CN disclosed
WO-1994014777-A1 HETEROCYCLIC CARBONIC ACID DERIVATIVES WHICH BIND TO RETINOID RECEPTORS (RAR) EISAI CO., LTD. (JP) 1994-07-07 WO disclosed